SCHEMBL8669728

SCHEMBL8669728

Cc1cc2ccc(Br)cc2nc1-n1cncn1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5AP P20292 4/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
BACE1 P56817 2/20 0.36
HTT P42858 2/20 0.34
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
LMNA P02545 1/20 0.34
POLB P06746 1/20 0.34
MAPT P10636 1/20 0.34
HPGD P15428 1/20 0.34
TSHR P16473 1/20 0.34
HSD17B10 Q99714 1/20 0.34
ADORA2A P29274 1/20 0.34
ADORA1 P30542 1/20 0.34
PDE10A Q9Y233 1/20 0.32
CYP1A2 P05177 3/20 0.32
CYP2C19 P33261 3/20 0.32
TDP1 Q9NUW8 1/20 0.32
CYP2C9 P11712 3/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8672242 0.83 APOBEC3A (0.37) ALOX5APMEN1KMT2AHTTKDM4E
SCHEMBL8671760 0.81 TDP1 (0.45) MEN1KMT2AHTTKDM4EALDH1A1
SCHEMBL8674069 0.81 MEN1 (0.34) ALOX5APMEN1KMT2AHTTKDM4E
SCHEMBL18057354 0.73 CASP3 (0.38) ALOX5APMEN1KMT2AHTTKDM4E
SCHEMBL20335460 0.72 L3MBTL1 (0.43) MEN1KMT2AKDM4EALDH1A1POLB
SCHEMBL9730644 0.70 KCNJ5 (0.37) ALOX5APKDM4EALDH1A1POLBMAPT
SCHEMBL11873901 0.69 TDP1 (0.62) MEN1KMT2ABACE1HTTKDM4E
SCHEMBL4364664 0.68 ADORA2A (0.42) ALOX5APKMT2AHTTKDM4EALDH1A1
SCHEMBL25323103 0.66 BACE1 (0.46) BACE1HTTKDM4EALDH1A1HSD17B10
SCHEMBL15448564 0.66 BACE1 (0.46) MEN1KMT2ABACE1HTTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5830903-A ANTIULCER AGENTS ALKALOIDA CHEMICAL CO., LTD. (HU) 1998-11-03 US disclosed
EP-0643579-A1 TRIAZOLE SUBSTITUTED QUINOLINE DERIVATIVES ALKALOIDA VEGYESZETI GYAR RT (HU) 1995-03-22 EP disclosed
WO-1994022413-A2 TRIAZOLE SUBSTITUTED QUINOLINE DERIVATIVES ALKALOIDA VEGYÉSZETI GYÁR RT. (HU) 1994-10-13 WO disclosed