SCHEMBL8669880

SCHEMBL8669880

O=C(O)CN1CCN(CCOCCOCCO)CCN(CC(=O)O)CCN(CC(=O)O)CC1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 1/20 0.43
ABCB11 O95342 1/20 0.42
CHRM2 P08172 1/20 0.42
ADRA2A P08913 1/20 0.42
DRD2 P14416 1/20 0.42
ADRA2B P18089 1/20 0.42
ADRA2C P18825 1/20 0.42
DRD4 P21917 1/20 0.42
HRH2 P25021 1/20 0.42
HTR2A P28223 1/20 0.42
HTR7 P34969 1/20 0.42
ADRA1A P35348 1/20 0.42
HRH1 P35367 1/20 0.42
DRD3 P35462 1/20 0.42
OPRK1 P41145 1/20 0.42
HTR2B P41595 1/20 0.42
HTR5A P47898 1/20 0.42
HTR6 P50406 1/20 0.42
KCNH2 Q12809 1/20 0.42
USP2 O75604 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8669650 0.98 HTR1A (0.44) HTR1AABCB11CHRM2ADRA2ADRD2
SCHEMBL25729443 0.98 HTR1A (0.44) HTR1AABCB11CHRM2ADRA2ADRD2
SCHEMBL31305373 0.84 MEN1 (0.55) HTR1AABCB11CHRM2ADRA2ADRD2
SCHEMBL31305372 0.84 MEN1 (0.55) HTR1AABCB11CHRM2ADRA2ADRD2
SCHEMBL8562841 0.84 HSD11B1 (0.40) HSD17B10MEN1KMT2AKDM4EALDH1A1
SCHEMBL4905012 0.82 HTR1A (0.54) HTR1AABCB11CHRM2ADRA2ADRD2
SCHEMBL8966405 0.82
SCHEMBL15435923 0.82 NAMPT (0.43) HTR1AABCB11CHRM2ADRA2ADRD2
SCHEMBL22266254 0.82 KDM4E (0.44) HTR1AABCB11CHRM2ADRA2ADRD2
SCHEMBL3553321 0.80 NAMPT (0.44) HTR1AABCB11CHRM2ADRA2ADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2833766-B2 1998-12-09 JP claimed
EP-0466200-B1 Aminocarboxylic acids and derivatives thereof NYCOMED IMAGING AS (NO) 1996-04-24 EP claimed
US-5419893-A Aminopolycarboxylic acids and derivatives thereof for magnetic resonance imaging NYCOMED IMAGING AS (NO) 1995-05-30 US claimed
EP-0466200-A1 Aminocarboxylic acids and derivatives thereof NYCOMED IMAGING AS (NO) 1992-01-15 EP claimed
WO-1989000557-A1 AMINOPOLYCARBOXYLIC ACIDS AND DERIVATIVES THEREOF COCKBAIN, JULIAN, RODERICK, MICHAELSON (GB) 1989-01-26 WO claimed
US-5531978-A CHELATE COMPOUNDS, IMAGING NYCOMED IMAGING AS (NO) 1996-07-02 US disclosed
EP-0466200-B1 Aminocarboxylic acids and derivatives thereof NYCOMED IMAGING AS (NO) 1996-04-24 EP disclosed
US-5419893-A Aminopolycarboxylic acids and derivatives thereof for magnetic resonance imaging NYCOMED IMAGING AS (NO) 1995-05-30 US disclosed
US-5198208-A Chelate compounds for diagnosis by magnetic resonance imaging, ultrasound or radiation therapy NYCOMED IMAGING AS (NO) 1993-03-30 US disclosed
EP-0466200-A1 Aminocarboxylic acids and derivatives thereof NYCOMED IMAGING AS (NO) 1992-01-15 EP disclosed
WO-1989000557-A1 AMINOPOLYCARBOXYLIC ACIDS AND DERIVATIVES THEREOF COCKBAIN, JULIAN, RODERICK, MICHAELSON (GB) 1989-01-26 WO disclosed