SCHEMBL8674372

SCHEMBL8674372

CCCCc1ccccc1-c1c(C(N)=O)cccc1C(=O)O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MYC P01106 1/20 0.44
KEAP1 Q14145 1/20 0.43
NFE2L2 Q16236 1/20 0.43
LTB4R2 Q9NPC1 1/20 0.42
BID P55957 3/20 0.42
MCL1 Q07820 3/20 0.42
BCL2L1 Q07817 2/20 0.42
BAK1 Q16611 2/20 0.42
KAT8 Q9H7Z6 2/20 0.42
LMNA P02545 2/20 0.42
MAPT P10636 2/20 0.42
FOLH1 Q04609 1/20 0.42
MEN1 O00255 1/20 0.42
NR1I2 O75469 1/20 0.42
CHRM2 P08172 1/20 0.42
CYP3A4 P08684 1/20 0.42
ADRA2A P08913 1/20 0.42
OPRK1 P41145 1/20 0.42
HTR2B P41595 1/20 0.42
SLC6A3 Q01959 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8674378 0.85 BID (0.46) MYCBIDMCL1BCL2L1BAK1
SCHEMBL27892555 0.84 SMN1; SMN2 (0.45) LTB4R2BIDMCL1BCL2L1BAK1
SCHEMBL28342495 0.83 CYP3A4 (0.48) KEAP1NFE2L2LTB4R2LMNAMAPT
SCHEMBL27547212 0.82 LMNA (0.44) KEAP1NFE2L2LTB4R2BIDMCL1
SCHEMBL25181813 0.81 FOLH1 (0.53) LTB4R2BIDMCL1BCL2L1BAK1
Benzene SCHEMBL28299279 0.81 KMT2A (0.51) LTB4R2BIDMCL1BCL2L1BAK1
SCHEMBL38662910 0.80 BID (0.52) BIDMCL1BCL2L1BAK1KAT8
SCHEMBL3706715 0.80 BID (0.52) BIDMCL1BCL2L1BAK1KAT8
SCHEMBL1002853 0.79 MAPT (0.53) LTB4R2BIDMCL1BCL2L1BAK1
SCHEMBL1513987 0.79 HNF4A (0.53) BIDMCL1BCL2L1BAK1KAT8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0862555-A1 SUBSTITUTED ARYL OR HETEROARYLAMIDES HAVING RETINOID-LIKE BIOLOGICAL ACTIVITY Allergan (US) 1998-09-09 EP disclosed
WO-1997019062-A1 SUBSTITUTED ARYL OR HETEROARYLAMIDES HAVING RETINOID-LIKE BIOLOGICAL ACTIVITY ALLERGAN (US) 1997-05-29 WO disclosed