SCHEMBL8679202

SCHEMBL8679202

C#CCn1c(-c2ccccc2)nc(CC)c(COCC)c1=O

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.39
CYP2C9 P11712 2/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2C19 P33261 1/20 0.38
TLR7 Q9NYK1 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.37
ALDH1A1 P00352 5/20 0.36
HSD17B10 Q99714 4/20 0.36
HPGD P15428 3/20 0.36
ADORA2A P29274 1/20 0.36
LMNA P02545 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
PTBP1 P26599 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
ADORA3 P0DMS8 1/20 0.35
KDM5A P29375 1/20 0.35
MAPK1 P28482 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8678382 0.88 TLR7 (0.43) KDM4ECYP2C9CYP1A2CYP2C19TLR7
SCHEMBL8678404 0.85 GCGR (0.43) KDM4ECYP2C9CYP1A2CYP2C19TLR7
SCHEMBL8680399 0.83 GCGR (0.39) KDM4ECYP2C9CYP1A2CYP2C19TLR7
SCHEMBL8676900 0.83 L3MBTL1 (0.43) KDM4ECYP2C9CYP1A2CYP2C19TLR7
SCHEMBL8677290 0.82 TLR7 (0.43) KDM4ECYP2C9CYP1A2CYP2C19TLR7
SCHEMBL8678398 0.81 KDM4E (0.44) KDM4ECYP2C9CYP1A2CYP2C19L3MBTL1
SCHEMBL8678204 0.81 CYP1A2 (0.38) KDM4ECYP2C9CYP1A2CYP2C19TLR7
SCHEMBL8676990 0.80 SMN1; SMN2 (0.41) KDM4ECYP2C9CYP1A2CYP2C19TLR7
SCHEMBL8678115 0.80 TLR7 (0.40) KDM4ECYP2C9TLR7L3MBTL1ALDH1A1
SCHEMBL8678090 0.80 TLR7 (0.42) KDM4ECYP2C9CYP1A2CYP2C19TLR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5726124-A IN MIXTURE WITH OTHER HERBICIDES, ALKYLATION AND ETHERIFICATION OF PYRIMIDINONE AND THIOPYRIMIDINONE COMPOUNDS ROHM AND HAAS COMPANY (US) 1998-03-10 US disclosed
CN-1109879-A 2-arylpyrimidines and herbicidal use thereof ROHM & HAAS (US) 1995-10-11 CN disclosed
EP-0663396-A1 2-Arylpyrimidines and herbicidal use thereof ROHM AND HAAS COMPANY (US) 1995-07-19 EP disclosed