SCHEMBL8679222

SCHEMBL8679222

O=C(NC(=O)c1c(F)cccc1F)Nc1nc2cc(Cl)ccc2s1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.60
RAB9A P51151 4/20 0.56
NPC1 O15118 3/20 0.56
MEN1 O00255 3/20 0.56
KMT2A Q03164 3/20 0.56
GHSR Q92847 2/20 0.52
PKM P14618 1/20 0.49
ALDH1A1 P00352 1/20 0.49
LMNA P02545 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
DHODH Q02127 1/20 0.48
DYRK1A Q13627 2/20 0.48
IDO1 P14902 1/20 0.47
PCSK9 Q8NBP7 1/20 0.47
HSD17B1 P14061 1/20 0.47
HSD17B2 P37059 1/20 0.47
RECQL P46063 1/20 0.46
LRRK2 Q5S007 1/20 0.46
FSCN1 Q16658 1/20 0.45
CASP3 P42574 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4912973 0.88 MAPT (0.74) MAPTRAB9ANPC1MEN1KMT2A
SCHEMBL2681868 0.84 RAB9A (0.68) MAPTRAB9ANPC1MEN1KMT2A
SCHEMBL4914400 0.83 MAPT (0.73) MAPTRAB9ANPC1MEN1KMT2A
SCHEMBL10736618 0.81 SMN1; SMN2 (0.68) MAPTRAB9ANPC1MEN1KMT2A
SCHEMBL11663113 0.79 GHSR (0.74) MAPTRAB9ANPC1MEN1KMT2A
SCHEMBL2242446 0.77 MAPT (0.75) MAPTRAB9ANPC1MEN1KMT2A
SCHEMBL11716373 0.77 MAPT (0.59) MAPTRAB9ANPC1GHSRSMN1; SMN2
SCHEMBL1785607 0.76 RAB9A (0.71) MAPTRAB9ANPC1MEN1KMT2A
SCHEMBL18851598 0.75 KDM4E (0.63) MAPTRAB9ANPC1MEN1KMT2A
SCHEMBL5097268 0.75 LRRK2 (0.73) RAB9ANPC1MEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5776981-A Use of acyl urea compounds for controlling endoparasites and ectoparasites of warm-blooded animals NOVARTIS CORPORATION (US) 1998-07-07 US disclosed
US-5776982-A Use of acyl urea compounds for controlling endoparasites and ectoparasites of warm-blooded animals NOVARTIS CORPORATION (US) 1998-07-07 US disclosed
US-5420163-A Insecticides or miticides CIBA-GEIGY (US) 1995-05-30 US disclosed
US-5135953-A Oral or injections; cattle, swine, poultry CIBA-GEIGY (US) 1992-08-04 US disclosed
EP-0211004-A1 USE OF ACYL UREA COMPOUNDS FOR CONTROLLING ENDOPARASITES AND ECTOPARASITES OF WARM-BLOODED ANIMALS RHONE-POULENC NEDERLAND B.V. (NL) 1987-02-25 EP disclosed
WO-1986003941-A1 USE OF ACYL UREA COMPOUNDS FOR CONTROLLING ENDOPARASITES AND ECTOPARASITES OF WARM-BLOODED ANIMALS UNION CARBIDE CORPORATION (US) 1986-07-17 WO disclosed