SCHEMBL8679335

SCHEMBL8679335

CC(O)C#Cc1ccc2cc(O)ccc2c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.41
TTR P02766 1/20 0.39
ESR1 P03372 6/20 0.38
ESR2 Q92731 6/20 0.38
CYP3A4 P08684 2/20 0.38
ALOX15 P16050 1/20 0.38
TSHR P16473 1/20 0.38
HIF1A Q16665 1/20 0.38
HSD17B10 Q99714 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
HCAR2 Q8TDS4 1/20 0.37
GABRP O00591 1/20 0.36
GABRD O14764 1/20 0.36
GABRA1 P14867 1/20 0.36
GABRB1 P18505 1/20 0.36
GABRG2 P18507 1/20 0.36
GABRB3 P28472 1/20 0.36
GABRA5 P31644 1/20 0.36
GABRA3 P34903 1/20 0.36
GABRA2 P47869 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5604749 0.81 APP (0.47) ESR1ESR2CYP3A4ALOX15HIF1A
SCHEMBL21741209 0.80 CYP1A2 (0.54) CYP1A2TTRESR1ESR2CYP3A4
SCHEMBL8679613 0.79 ABCB11 (0.45) CYP1A2TSHRTDP1APPCYP2D6
SCHEMBL21967023 0.78 CYP1A2 (0.52) CYP1A2TTRESR1ESR2CYP3A4
SCHEMBL3216361 0.78 APP (0.38) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL22750625 0.77 CYP1A2 (0.52) CYP1A2TTRESR1ESR2CYP3A4
SCHEMBL29946581 0.77 CYP1A2 (0.52) CYP1A2TTRESR1ESR2CYP3A4
SCHEMBL8517544 0.73 ALDH1A1 (0.41) CYP3A4ALOX15TSHRTDP1GABRA1
SCHEMBL2473384 0.73 CYP1A2 (0.42) CYP1A2TTRESR1ESR2CYP3A4
SCHEMBL21836123 0.72 ASIC3 (0.57) CYP1A2ESR1ESR2CYP3A4ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998024747-A1 A PROCESS FOR THE PREPARATION OF NABUMETONE RECORDATI S.A. CHEMICAL AND PHARMACEUTICAL COMPANY (CH) 1998-06-11 WO claimed
WO-1998024747-A1 A PROCESS FOR THE PREPARATION OF NABUMETONE RECORDATI S.A. CHEMICAL AND PHARMACEUTICAL COMPANY (CH) 1998-06-11 WO disclosed