SCHEMBL8679771

SCHEMBL8679771

NC(=O)n1c(O)cc2ccccc21

nearest known ligand 0.49

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KDR P35968 13/20 0.49
PDGFRB P09619 10/20 0.49
DAO P14920 2/20 0.42
SLC9A1 P19634 1/20 0.41
MCL1 Q07820 1/20 0.41
ALDH1A1 P00352 1/20 0.40
TSHR P16473 1/20 0.40
CCR2 P41597 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27265492 0.98 KDR (0.48) KDRPDGFRBDAOSLC9A1MCL1
SCHEMBL4467286 0.82 DAO (0.47) KDRPDGFRBDAOMCL1ALDH1A1
SCHEMBL17022579 0.81 POLB (0.52) DAOSLC9A1MCL1ALDH1A1TSHR
SCHEMBL27308385 0.80 LDHA (0.51) KDRPDGFRBMCL1ALDH1A1CCR2
SCHEMBL31122079 0.79 KDR (0.51) KDRPDGFRBSLC9A1MCL1ALDH1A1
SCHEMBL27597857 0.79 KDR (0.51) KDRPDGFRBDAOSLC9A1MCL1
SCHEMBL8360588 0.79 KDR (0.51) KDRPDGFRBSLC9A1MCL1ALDH1A1
SCHEMBL17022686 0.78 SRC (0.53) DAOMCL1TSHR
Benzene SCHEMBL28136154 0.78 KDR (0.50) KDRPDGFRBDAOSLC9A1MCL1
Hydrochloric Acid SCHEMBL28136871 0.78 KDR (0.50) KDRPDGFRBSLC9A1MCL1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 24 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1093704-A Regioselective synthesis of 4-chloro-2-thiophenecarboxylic acid PFIZER (US) 1994-10-19 CN claimed
CN-85103527-A Preparation N, the method for the disubstituted 2-hydroxyindole of 3--1-hydroxyalkyl cooh amide 1987-01-28 CN claimed
JP-10087614-A None JP disclosed
JP-4235165-A None JP disclosed
JP-H1087614-A STABLE AND LONG-TIME ACTING SALT OF CARBOXAMIDE FOR CURING ARTICULAR DISEASE PFIZER INC 1998-04-07 JP disclosed
WO-1997022605-A1 STABLE, LONG ACTING SALTS OF INDOLE DERIVATIVES FOR THE TREATMENT OF JOINT DISEASES PFIZER INC. (US) 1997-06-26 WO disclosed
CN-1136921-A Pharmaceutical agents for treatment of alzheimer's disease PFIZER (US) 1996-12-04 CN disclosed
CN-1123144-A 3-substituted-2-oxindoles as inhibitors of viral replication PFIZER (US) 1996-05-29 CN disclosed
CN-1099614-A 6-chloro-5-fluoro-3-(2-thenoyl)-2-oxindole-1-carboxamide as an analgesic and anti-inflammatory agent PFIZER (US) 1995-03-08 CN disclosed
CN-1093704-A Regioselective synthesis of 4-chloro-2-thiophenecarboxylic acid PFIZER (US) 1994-10-19 CN disclosed
CN-1022324-C Anhydrous crystal sodium salt of 5-chloro-3-(2-thenoyl)-2-oxyindole-1-carboxamide PFIZER (US) 1993-10-06 CN disclosed
CN-1003855-B Process for preparing 1, 3-disubstituted 2-oxindoles 美国辉瑞有限公司 1989-04-12 CN disclosed
CN-1003855-B Process for preparing 1, 3-disubstituted 2-oxindoles 美国辉瑞有限公司 1989-04-12 CN disclosed
CN-88100555-A Anhydrous, crystalline sodium salt of 5-chloro-3- (2-thenoyl) -2-hydroxyindole-1-carboxamide 1988-08-17 CN disclosed
CN-85101795-A With 1, the two 2-oxyindoles that replace of 3-prepare pain killer and antiphlogistic 1987-04-08 CN disclosed
CN-85103527-A Preparation N, the method for the disubstituted 2-hydroxyindole of 3--1-hydroxyalkyl cooh amide 1987-01-28 CN disclosed
CN-85103527-A Preparation N, the method for the disubstituted 2-hydroxyindole of 3--1-hydroxyalkyl cooh amide 1987-01-28 CN disclosed
CN-85101029-A The method of preparation-2-oxyindole-1-methane amide and intermediate product thereof 1987-01-24 CN disclosed
CN-85101028-A Be used as the preparation of 2-oxyindole-1-methane amide that the 3-of anodyne and antiphlogistic replaces 1987-01-17 CN disclosed
CN-85101028-A Be used as the preparation of 2-oxyindole-1-methane amide that the 3-of anodyne and antiphlogistic replaces 1987-01-17 CN disclosed