SCHEMBL868087

SCHEMBL868087

OC(CC1CC1)c1ccc(Cl)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AOC3 Q16853 1/20 0.46
GRIN1 Q05586 5/20 0.44
GRIN2B Q13224 5/20 0.44
GMNN O75496 1/20 0.44
TP53 P04637 1/20 0.44
CYP3A4 P08684 1/20 0.44
ALOX15 P16050 1/20 0.44
TSHR P16473 1/20 0.44
NFKB1 P19838 1/20 0.44
THPO P40225 1/20 0.44
MTOR P42345 1/20 0.44
BLM P54132 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
SLC6A2 P23975 2/20 0.44
SLC6A4 P31645 2/20 0.44
SLC6A3 Q01959 2/20 0.44
FFAR2 O15552 1/20 0.42
GRIN2D O15399 4/20 0.41
GRIN3B O60391 4/20 0.41
GRIN2A Q12879 4/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10633563 0.91 SLC6A2 (0.54) AOC3GRIN1GRIN2BGMNNTP53
SCHEMBL13391312 0.88 SLC6A2 (0.46) AOC3GRIN1GRIN2BGMNNTP53
Hydrochloric Acid SCHEMBL15535999 0.86 SLC6A2 (0.48) GRIN1GRIN2BGMNNTP53CYP3A4
SCHEMBL15535932 0.81 TP53 (0.44) GRIN1GRIN2BGMNNTP53CYP3A4
SCHEMBL23536506 0.80 SLC18A3 (0.45)
SCHEMBL17609122 0.80 SLC18A3 (0.45)
SCHEMBL13308375 0.79 SLC18A3 (0.47) SLC6A2SLC6A4SLC6A3
SCHEMBL16622109 0.79 CYP1A2 (0.58) AOC3
SCHEMBL16622110 0.79 CYP1A2 (0.58) AOC3
SCHEMBL13741859 0.79 CYP1A2 (0.58) AOC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 19 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106883266-B Preparation method of 1- (4-chlorphenyl) -2-cyclopropyl-1-acetone and intermediate thereof 江苏七洲绿色化工股份有限公司 2020-03-17 CN disclosed
CN-103044230-B Preparation method of 1-(4-chlorphenyl)-2-cyclopropyl-1-acetone HUNAN CHEMICAL ENGINEERING INST. (CN) 2014-10-08 CN disclosed
CN-102584558-B Preparation method of 1-(4-chlorphenyl)-2-cyclopropyl-1-acetone HUNAN RES INST CHEMICAL IND 2013-10-30 CN disclosed
CN-103044230-A Preparation method of 1-(4-chlorphenyl)-2-cyclopropyl-1-acetone HUNAN RES INST CHEMICAL IND 2013-04-17 CN disclosed
CN-102584558-A Preparation method of 1-(4-chlorphenyl)-2-cyclopropyl-1-acetone HUNAN RES INST CHEMICAL IND 2012-07-18 CN disclosed
EP-2440535-A1 ANTIFUNGAL 1,2,4-TRIAZOLYL DERIVATIVES HAVING A 5- SULFUR SUBSTITUENT BASF SE (DE) 2012-04-18 EP disclosed
US-20120077676-A1 Antifungal 1,2,4-Triazolyl Derivatives Having a 5-Sulfur Substituent BASF SE (DE) 2012-03-29 US disclosed
WO-2010142779-A1 ANTIFUNGAL 1,2,4-TRIAZOLYL DERIVATIVES HAVING A 5- SULFUR SUBSTITUENT BASF SE (DE) 2010-12-16 WO disclosed
EP-0900218-B1 HETEROCYCLIC COMPOUNDS LILLY CO ELI (US) 2002-07-24 EP disclosed
EP-0900218-A4 HETEROCYCLIC COMPOUNDS LILLY CO ELI (US) 2001-05-23 EP disclosed
US-6117883-A Heterocyclic compounds ELI LILLY AND COMPANY (US) 2000-09-12 US disclosed
EP-0900218-A1 HETEROCYCLIC COMPOUNDS ELI LILLY AND COMPANY (US) 1999-03-10 EP disclosed
CN-1041717-C Cyclopropane derivatives SANDOZ LTD (CH) 1999-01-20 CN disclosed
US-5770741-A FUNGICIDE INTERMEDIATE SANDOZ LTD. (CH) 1998-06-23 US disclosed
WO-1997040044-A1 HETEROCYCLIC COMPOUNDS ELI LILLY AND COMPANY (US) 1997-10-30 WO disclosed
EP-0321409-B1 CYCLOPROPANE DERIVATIVES SANDOZ AG (CH) 1993-03-17 EP disclosed
US-4973767-A SUBSTITUTED ETHANOLS, CHEMICAL INTERMEDIATES FOR FUNGICIDES SANDOZ LTD. (CH) 1990-11-27 US disclosed
CN-1035494-A The preparation method of cyclopropane derivative SANDOZ LTD (CH) 1989-09-13 CN disclosed
EP-0321409-A2 Cyclopropane derivatives SANDOZ AG (CH) 1989-06-21 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120077676-A1 Antifungal 1,2,4-Triazolyl Derivatives Having a 5-Sulfur Substituent ERG28, STS, CYP51A1 AOC3 357/4885GRIN1 1668/4885GRIN2B 2208/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.