SCHEMBL8682011

SCHEMBL8682011

Cc1cccc(Cl)c1NC(N)=O

nearest known ligand 0.60

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.60
PDK1 Q15118 1/20 0.56
PDK2 Q15119 1/20 0.56
PDK3 Q15120 1/20 0.56
PDK4 Q16654 1/20 0.56
CHRNA7 P36544 10/20 0.49
MAPK14 Q16539 1/20 0.48
DRD2 P14416 1/20 0.47
HTR2A P28223 1/20 0.47
HTR2B P41595 1/20 0.47
ALDH1A1 P00352 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
MAOB P27338 1/20 0.47
CXCL8 P10145 1/20 0.47
PTGS2 P35354 1/20 0.47
PKM P14618 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5520683 0.86 DRD2 (0.59) GAADRD2HTR2AHTR2BALDH1A1
SCHEMBL1439894 0.86 TYK2 (0.52) GAAPDK1PDK2PDK3PDK4
SCHEMBL11402399 0.85 PDK1 (0.59) GAAPDK1PDK2PDK3PDK4
SCHEMBL4099006 0.84 GAA (0.51) GAAPDK1PDK2PDK3PDK4
SCHEMBL2921682 0.83 PDK1 (0.58) GAAPDK1PDK2PDK3PDK4
SCHEMBL9037897 0.82 GAA (0.66) GAAPDK1PDK2PDK3PDK4
SCHEMBL11735899 0.81 PDK1 (0.56) GAAPDK1PDK2PDK3PDK4
Hydrochloric Acid SCHEMBL9004815 0.81 GAA (0.64) GAAPDK1PDK2PDK3PDK4
SCHEMBL7168272 0.80 DRD2 (0.55) GAAPDK1PDK2PDK3PDK4
SCHEMBL14889779 0.79 POLB (0.56) GAADRD2HTR2AHTR2BALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114867525-A Dihydrocyclopentaisoquinoline derivatives UCB生物制药有限责任公司 2022-08-05 CN claimed
CN-114867525-A Dihydrocyclopentaisoquinoline derivatives UCB生物制药有限责任公司 2022-08-05 CN disclosed
US-5780483-A IL-8 receptor antagonists SMITHKLINE BEECHAM CORPORATION (US) 1998-07-14 US disclosed
EP-0182166-B1 PROCESS FOR PREPARING PHENYLISOPROPYLUREA COMPOUNDS AMERICAN CYANAMID COMPANY (US) 1989-05-31 EP disclosed
US-4578513-A Process for preparing phenylisopropylurea compounds AMERICAN CYANAMID COMPANY (US) 1986-03-25 US disclosed