SCHEMBL8683058

SCHEMBL8683058

CCCC#CN1CC(=O)CC(c2cccc3ccccc23)=N1

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 2/20 0.32
CNR1 P21554 2/20 0.32
CNR2 P34972 2/20 0.32
BCHE P06276 1/20 0.32
TLR8 Q9NR97 1/20 0.32
KDM4E B2RXH2 2/20 0.32
ALDH1A1 P00352 1/20 0.32
LMNA P02545 1/20 0.32
HPGD P15428 1/20 0.32
ALPL P05186 1/20 0.32
GAA P10253 1/20 0.32
GSK3A P49840 1/20 0.31
GSK3B P49841 1/20 0.31
BRD4 O60885 1/20 0.31
CREBBP Q92793 1/20 0.31
PARP1 P09874 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8301456 0.84 KIF11 (0.36)
SCHEMBL8301250 0.84 KIF11 (0.36) ALDH1A1LMNAHPGD
SCHEMBL8683206 0.81 ALDH1A1 (0.35) ALDH1A1HPGDCREBBP
SCHEMBL8300278 0.76 CHRNB4 (0.34) TLR8ALDH1A1
SCHEMBL8300862 0.69 PTGS1 (0.33)
SCHEMBL8302889 0.65 KIF11 (0.38) BCHEKDM4EALDH1A1LMNAGAA
SCHEMBL8684712 0.64 KCNH2 (0.32) KDM4EALDH1A1LMNAGAA
SCHEMBL8683056 0.63 LMNA (0.37) KDM4EALDH1A1LMNAHPGDALPL
SCHEMBL18654341 0.60 NISCH (0.46) KDM4EALDH1A1HPGDALPLGAA
SCHEMBL1612398 0.58 TLR8 (0.50) TLR8KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753642-A AGRICULTURE, MEDICINE ROHM AND HAAS COMPANY (US) 1998-05-19 US disclosed
US-5728715-A FOR MAMMALS, AGRICULTURE, RICE, WHEAT, TOMATOES ROHM AND HAAS COMPANY (US) 1998-03-17 US disclosed
US-5728694-A Dihydropyridazinones, pyridazinones and related compounds as fungicides ROHM AND HAAS COMPANY (US) 1998-03-17 US disclosed
US-5728698-A AGRICULTURAL USE, RICE, WHEAT ROHM AND HAAS COMPANY (US) 1998-03-17 US disclosed
US-5726176-A FOR CONTROLLING AGRICULTURAL AND MAMMALIAN FUNGAL DISEASES ROHM AND HAAS COMPANY (US) 1998-03-10 US disclosed
US-5726162-A FOR CONTROLLING AGRICULTURAL AND MAMMALIAN FUNGAL DISEASES ROHM AND HAAS COMPANY (US) 1998-03-10 US disclosed
US-5631254-A RICE; HUMAN INFECTIONS ROHM AND HAAS COMPANY (US) 1997-05-20 US disclosed
US-5552409-A PHYTOPATHOGENIC, RICE ROHM AND HAAS COMPANY (US) 1996-09-03 US disclosed
EP-0478195-A1 Dihydropyridazinones, pyridazinones and related compounds as fungicides ROHM AND HAAS COMPANY (US) 1992-04-01 EP disclosed