SCHEMBL8683096

SCHEMBL8683096

CCCC#CN1CC(=O)CC(c2ccccc2OC)=N1

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PDCD1 Q15116 1/20 0.46
CD274 Q9NZQ7 1/20 0.46
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
UGCG Q16739 6/20 0.35
ADORA3 P0DMS8 2/20 0.35
ADORA1 P30542 2/20 0.35
KDM4E B2RXH2 2/20 0.35
ALDH1A1 P00352 1/20 0.35
DRD2 P14416 1/20 0.35
DRD4 P21917 1/20 0.35
DRD3 P35462 1/20 0.35
CRBN Q96SW2 1/20 0.34
NPC1 O15118 1/20 0.33
CA12 O43570 1/20 0.33
RAB9A P51151 1/20 0.33
TLR8 Q9NR97 1/20 0.33
HSD17B10 Q99714 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8685396 0.87 KIF11 (0.34) PDCD1CD274
SCHEMBL8301456 0.84 KIF11 (0.36) ADORA3ADORA1CRBN
SCHEMBL8301250 0.84 KIF11 (0.36) PDCD1CD274MEN1KMT2AALDH1A1
SCHEMBL8683206 0.77 ALDH1A1 (0.35) ALDH1A1DRD2HSD17B10
SCHEMBL8685267 0.76 BTK (0.37) PDCD1CD274ALDH1A1NPC1
SCHEMBL8683364 0.76 NPC1 (0.32) NPC1RAB9A
SCHEMBL8683453 0.74 RAB9A (0.36) MEN1KMT2AKDM4EALDH1A1NPC1
SCHEMBL8300278 0.74 CHRNB4 (0.34) ALDH1A1TLR8
SCHEMBL8683436 0.73 NPC1 (0.36) MEN1KMT2AKDM4EALDH1A1NPC1
SCHEMBL8304845 0.73 KIF11 (0.37) MEN1KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753642-A AGRICULTURE, MEDICINE ROHM AND HAAS COMPANY (US) 1998-05-19 US disclosed
US-5728694-A Dihydropyridazinones, pyridazinones and related compounds as fungicides ROHM AND HAAS COMPANY (US) 1998-03-17 US disclosed
US-5728715-A FOR MAMMALS, AGRICULTURE, RICE, WHEAT, TOMATOES ROHM AND HAAS COMPANY (US) 1998-03-17 US disclosed
US-5728698-A AGRICULTURAL USE, RICE, WHEAT ROHM AND HAAS COMPANY (US) 1998-03-17 US disclosed
US-5726176-A FOR CONTROLLING AGRICULTURAL AND MAMMALIAN FUNGAL DISEASES ROHM AND HAAS COMPANY (US) 1998-03-10 US disclosed
US-5726162-A FOR CONTROLLING AGRICULTURAL AND MAMMALIAN FUNGAL DISEASES ROHM AND HAAS COMPANY (US) 1998-03-10 US disclosed
US-5631254-A RICE; HUMAN INFECTIONS ROHM AND HAAS COMPANY (US) 1997-05-20 US disclosed
US-5552409-A PHYTOPATHOGENIC, RICE ROHM AND HAAS COMPANY (US) 1996-09-03 US disclosed
EP-0478195-A1 Dihydropyridazinones, pyridazinones and related compounds as fungicides ROHM AND HAAS COMPANY (US) 1992-04-01 EP disclosed