SCHEMBL8685397

SCHEMBL8685397

NC(=S)NN=Cc1cc(N(CCO)CCO)ccn1

nearest known ligand 0.52

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
RRM2 P31350 8/20 0.45
NCOA3 Q9Y6Q9 2/20 0.41
RRM1 P23921 1/20 0.41
RRM2B Q7LG56 1/20 0.41
CISD1 Q9NZ45 1/20 0.41
KDM4E B2RXH2 1/20 0.41
POLB P06746 1/20 0.40
NCOA1 Q15788 1/20 0.40
MAOA P21397 1/20 0.40
MAOB P27338 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8688249 0.82 MAOA (0.57) RRM2NCOA3RRM1RRM2BCISD1
SCHEMBL293101 0.69 TOP2A (0.68) RRM2NCOA3RRM1RRM2BCISD1
SCHEMBL534248 0.69 TOP2A (0.68) RRM2NCOA3RRM1RRM2BCISD1
SCHEMBL8683198 0.68 RRM2 (0.43) RRM2NCOA3RRM1RRM2BCISD1
SCHEMBL8683949 0.67 RRM2 (0.44) RRM2NCOA3RRM1RRM2BCISD1
SCHEMBL17835748 0.65 RRM2 (0.55) RRM2NCOA3RRM1RRM2BCISD1
SCHEMBL17835747 0.65 RRM2 (0.55) RRM2NCOA3RRM1RRM2BCISD1
SCHEMBL13826735 0.64 POLB (0.61) RRM2KDM4EPOLBMAOB
SCHEMBL17835729 0.63 POLB (0.59) KDM4EPOLBMAOAMAOB
SCHEMBL17835730 0.63 POLB (0.59) KDM4EPOLBMAOAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5721259-A Method of using 2-formylpyridine thiosemicarbazone compounds YALE UNIVERSITY (US) 1998-02-24 US disclosed
EP-0570294-B1 2-Formylpyridine thiosemicarbazone derivatives, their preparation and their use as antitumor agents UNIV YALE (US) 1997-07-30 EP disclosed
US-5281715-A 2-formylpyridine thiosemicarbazone compounds YALE UNIVERSITY (US) 1994-01-25 US disclosed
EP-0570294-A1 2-Formylpyridine thiosemicarbazone derivatives, their preparation and their use as antitumor agents YALE UNIVERSITY (US) 1993-11-18 EP disclosed