SCHEMBL8683198

SCHEMBL8683198

NC(=S)NN=Cc1cc(N2CCCCC2)ccn1

nearest known ligand 0.52

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
RRM2 P31350 9/20 0.43
NCOA3 Q9Y6Q9 3/20 0.41
RRM1 P23921 1/20 0.41
RRM2B Q7LG56 1/20 0.41
CISD1 Q9NZ45 1/20 0.41
KDM4E B2RXH2 2/20 0.41
RAB9A P51151 1/20 0.41
POLB P06746 1/20 0.40
NCOA1 Q15788 2/20 0.40
HRH4 Q9H3N8 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8683949 0.79 RRM2 (0.44) RRM2NCOA3RRM1RRM2BCISD1
SCHEMBL28618179 0.74 KDM4E (0.67) KDM4EPOLB
SCHEMBL6167874 0.72 HRH4 (0.47) KDM4EHRH4
SCHEMBL6167866 0.72 HRH4 (0.47) KDM4EHRH4
SCHEMBL8688249 0.71 MAOA (0.57) RRM2NCOA3RRM1RRM2BCISD1
Hydrochloric Acid SCHEMBL7260368 0.71 HRH4 (0.46) KDM4EHRH4
Hydrochloric Acid SCHEMBL7260366 0.71 HRH4 (0.46) KDM4EHRH4
SCHEMBL534248 0.69 TOP2A (0.68) RRM2NCOA3RRM1RRM2BCISD1
SCHEMBL293101 0.69 TOP2A (0.68) RRM2NCOA3RRM1RRM2BCISD1
SCHEMBL25813337 0.69 HRH4 (0.47) KDM4EHRH4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5721259-A Method of using 2-formylpyridine thiosemicarbazone compounds YALE UNIVERSITY (US) 1998-02-24 US disclosed
EP-0570294-B1 2-Formylpyridine thiosemicarbazone derivatives, their preparation and their use as antitumor agents UNIV YALE (US) 1997-07-30 EP disclosed
US-5281715-A 2-formylpyridine thiosemicarbazone compounds YALE UNIVERSITY (US) 1994-01-25 US disclosed
EP-0570294-A1 2-Formylpyridine thiosemicarbazone derivatives, their preparation and their use as antitumor agents YALE UNIVERSITY (US) 1993-11-18 EP disclosed