SCHEMBL8686302

SCHEMBL8686302

COc1ccc(Nc2ncc(C(=O)O)cn2)cc1OC

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK8 P45983 1/20 0.57
MAPK9 P45984 1/20 0.57
FLT3 P36888 1/20 0.56
CA12 O43570 1/20 0.53
CA1 P00915 1/20 0.53
CA2 P00918 1/20 0.53
CA4 P22748 1/20 0.53
CA6 P23280 1/20 0.53
CA7 P43166 1/20 0.53
TPMT P51580 1/20 0.53
CA9 Q16790 1/20 0.53
CA14 Q9ULX7 1/20 0.53
HDAC3 O15379 2/20 0.50
HDAC1 Q13547 2/20 0.50
HDAC2 Q92769 2/20 0.50
HDAC6 Q9UBN7 2/20 0.50
MAPT P10636 3/20 0.48
CDK4 P11802 1/20 0.48
CCND1 P24385 1/20 0.48
CCND2 P30279 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8682666 0.89 MAPT (0.56) MAPK8MAPK9FLT3HDAC3HDAC1
SCHEMBL8686294 0.82 MAPK8 (0.54) MAPK8MAPK9FLT3CDK4CCND1
SCHEMBL3634270 0.81 HDAC3 (0.74) CA1CA2HDAC3HDAC1HDAC2
SCHEMBL8686297 0.78 L3MBTL1 (0.55) CA12CA1CA2CA4CA6
SCHEMBL5038697 0.76 MAPK13 (0.52) MAPK8MAPK9MAPTCTSVCTSL
SCHEMBL4489904 0.76 MAPK8 (0.48) MAPK8MAPK9FLT3HDAC3HDAC1
SCHEMBL3269159 0.74 ABCG2 (0.67) FLT3MAPTEGFRNPC1RAB9A
SCHEMBL4485439 0.74 SYK (0.59) MAPK8MAPK9FLT3HDAC3HDAC1
SCHEMBL14657966 0.73 MAPK8 (1.00) MAPK8MAPK9EGFRITK
SCHEMBL670354 0.73 HDAC6 (0.72) MAPK8HDAC3HDAC1HDAC2HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5719187-A Compounds having a guanidine structure and pharmaceutical composition containing same CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE(CNRS) (FR) 1998-02-17 US disclosed
US-5480884-A Compounds having a guanidine structure CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 1996-01-02 US disclosed