SCHEMBL8686933

SCHEMBL8686933

N#CCCC1CCCCN1Cc1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 1/20 0.53
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
OPRD1 P41143 1/20 0.47
SIGMAR1 Q99720 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8414528 0.96 SLC6A4 (0.48) SLC6A4MEN1KMT2A
SCHEMBL1257677 0.85 SLC6A4 (0.49) SLC6A4OPRD1
SCHEMBL1257675 0.85 SLC6A4 (0.49) SLC6A4OPRD1
SCHEMBL10682307 0.82 MEN1 (0.62) SLC6A4MEN1KMT2A
SCHEMBL5967865 0.82 OPRD1 (0.51) SLC6A4MEN1KMT2AOPRD1SIGMAR1
SCHEMBL11969174 0.82 OPRD1 (0.51) SLC6A4MEN1KMT2AOPRD1SIGMAR1
SCHEMBL11969306 0.81 SIGMAR1 (0.62) OPRD1SIGMAR1
SCHEMBL4331465 0.81 SIGMAR1 (0.62) OPRD1SIGMAR1
SCHEMBL13267225 0.81 OPRD1 (0.50) SLC6A4MEN1KMT2AOPRD1SIGMAR1
SCHEMBL11990438 0.81 OPRD1 (0.56) SLC6A4MEN1KMT2AOPRD1SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108409738-B 3, 4-methylenedioxyphenyl substituted tetrahydro-beta-carboline piperazine diketone derivative and application thereof 华东理工大学 2020-10-16 CN disclosed
US-5834499-A TREATING GASTROINTESTINAL DISORDERS YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1998-11-10 US disclosed
CN-1143364-A 5-HT3 receptor agonist, novel thiazole derivative, and intermediate thereof YAMANOUCHI PHARMA CO LTD (JP) 1997-02-19 CN disclosed
EP-0749966-A1 5-HT 3 RECEPTOR AGONIST, NOVEL THIAZOLE DERIVATIVE, AND INTERMEDIATE THEREFOR YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1996-12-27 EP disclosed