SCHEMBL8689243

SCHEMBL8689243

O=C(CBr)Nc1ccc(Br)cc1C(=O)O

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 3/20 0.68
KDM4E B2RXH2 2/20 0.68
POLB P06746 2/20 0.67
MEN1 O00255 6/20 0.58
KMT2A Q03164 6/20 0.58
APEX1 P27695 1/20 0.56
AKR1C2 P52895 2/20 0.55
AKR1C1 Q04828 2/20 0.55
AKR1C4 P17516 1/20 0.55
AKR1C3 P42330 1/20 0.55
MAPK1 P28482 2/20 0.52
ALDH1A1 P00352 3/20 0.51
MAPT P10636 2/20 0.51
PLA2G1B P04054 1/20 0.51
HPGD P15428 1/20 0.51
ATG4B Q9Y4P1 1/20 0.51
HTT P42858 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50
TRPM2 O94759 1/20 0.49
KCNK2 O95069 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29440123 0.87 TDP1 (0.73) TDP1KDM4EPOLBMEN1KMT2A
SCHEMBL140563 0.87 TDP1 (0.73) TDP1KDM4EPOLBMEN1KMT2A
SCHEMBL8688878 0.85 KMT2A (0.55) TDP1KDM4EPOLBMEN1KMT2A
SCHEMBL7532175 0.84 POLB (0.68) TDP1KDM4EPOLBMEN1KMT2A
SCHEMBL16650906 0.83 ALDH1A1 (0.60) TDP1KDM4EPOLBMEN1KMT2A
SCHEMBL8484239 0.82 KCNK2 (0.49) TDP1KDM4EPOLBALDH1A1MAPT
SCHEMBL8482804 0.82 KDM4E (0.64) KDM4EPOLBMEN1KMT2AAKR1C2
SCHEMBL15647380 0.81 KMT2A (0.67) TDP1KDM4EPOLBMEN1KMT2A
SCHEMBL6354673 0.81 NPC1 (0.59) TDP1KDM4EPOLBMEN1KMT2A
SCHEMBL16655841 0.80 KDM4E (0.68) TDP1KDM4EPOLBMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5741926-A ANTIDIABETIC AGENT SHAMAN PHARMACEUTICALS, INC. (US) 1998-04-21 US disclosed
WO-1997030019-A1 ANILINE DERIVATIVES HAVING ANTIHYPERGLYCEMIC ACTIVITY SHAMAN PHARMACEUTICALS, INC. (US) 1997-08-21 WO disclosed