SCHEMBL8690762

SCHEMBL8690762

COC(C)OCOc1ccc(C(=O)O)c(OC(=O)c2ccccc2)c1C12CC3CC(CC(C3)C1)C2

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 3/20 0.37
EPHX2 P34913 2/20 0.36
KDM4E B2RXH2 1/20 0.35
RARA P10276 3/20 0.34
HIF1A Q16665 6/20 0.33
EPAS1 Q99814 3/20 0.33
RARB P10826 2/20 0.33
RARG P13631 2/20 0.33
ESR1 P03372 1/20 0.33
ESR2 Q92731 1/20 0.33
MEN1 O00255 1/20 0.32
NR1I2 O75469 1/20 0.32
LMNA P02545 1/20 0.32
PGR P06401 1/20 0.32
HSPD1 P10809 1/20 0.32
GOT1 P17174 1/20 0.32
GLRA1 P23415 1/20 0.32
BLM P54132 1/20 0.32
HSPE1 P61604 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8691802 0.88 EPHX2 (0.35) IKBKBEPHX2RARAHIF1AEPAS1
SCHEMBL8691383 0.88 PTPN1 (0.41) IKBKBEPHX2RARAHIF1AEPAS1
SCHEMBL8397841 0.87 EPHX2 (0.35) IKBKBEPHX2KDM4ERARAHIF1A
SCHEMBL8568404 0.80 IKBKB (0.35) IKBKBEPHX2KDM4ERARAHIF1A
SCHEMBL8394738 0.77 HIF1A (0.36) IKBKBKDM4ERARAHIF1AEPAS1
SCHEMBL8574908 0.76 IKBKB (0.33) IKBKBRARAHIF1AEPAS1LMNA
SCHEMBL8575216 0.74 IKBKB (0.34) IKBKBEPHX2KDM4ERARAHIF1A
SCHEMBL8426205 0.74 RARA (0.51) IKBKBRARAHIF1AEPAS1RARB
SCHEMBL5888166 0.74 RARA (0.55) IKBKBKDM4ERARARARBRARG
SCHEMBL8692338 0.73 RARA (0.45) IKBKBRARARARBRARGMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5786379-A Adamantyl-substituted biaromatic compounds and pharmaceutical/cosmetic compositions comprised thereof CENTRE INTERNATIONAL DE RECHERCHES DERMATOLOGIQUES GALDERMA (FR) 1998-07-28 US claimed
US-5786379-A Adamantyl-substituted biaromatic compounds and pharmaceutical/cosmetic compositions comprised thereof CENTRE INTERNATIONAL DE RECHERCHES DERMATOLOGIQUES GALDERMA (FR) 1998-07-28 US disclosed