SCHEMBL8693185

SCHEMBL8693185

CCOC(=O)CCCn1c(C(=O)O)cc2ccccc21

nearest known ligand 0.58

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 4/20 0.58
ALDH1A1 P00352 1/20 0.56
CYP1A2 P05177 1/20 0.56
POLB P06746 1/20 0.56
TNF P01375 2/20 0.54
KDM4E B2RXH2 1/20 0.53
CRHBP P24387 1/20 0.53
CRHR2 Q13324 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
CCR2 P41597 2/20 0.52
MEN1 O00255 1/20 0.52
KMT2A Q03164 1/20 0.52
GAA P10253 1/20 0.51
CTNNB1 P35222 1/20 0.50
NOD2 Q9HC29 1/20 0.49
NOD1 Q9Y239 1/20 0.49
PTGDR2 Q9Y5Y4 3/20 0.48
CNR1 P21554 1/20 0.48
CNR2 P34972 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8691611 0.96 MCL1 (0.57) MCL1ALDH1A1CYP1A2POLBTNF
SCHEMBL7686010 0.95 MCL1 (0.56) MCL1ALDH1A1CYP1A2POLBTNF
SCHEMBL6701625 0.92 ALDH1A1 (0.59) MCL1ALDH1A1CYP1A2POLBKDM4E
SCHEMBL8653460 0.86 KDM4E (0.64) TNFKDM4ECRHBPCRHR2SMN1; SMN2
SCHEMBL7686434 0.86 PLA2G4A (0.46) MCL1ALDH1A1CYP1A2POLBTNF
SCHEMBL7256497 0.84 MEN1 (0.63) MCL1ALDH1A1CYP1A2POLBKDM4E
SCHEMBL2480710 0.84 ALDH1A1 (0.57) MCL1ALDH1A1CYP1A2POLBCCR2
SCHEMBL8689867 0.83 KDM4E (0.54) TNFKDM4ECRHBPCRHR2SMN1; SMN2
SCHEMBL2015584 0.83 SRD5A2 (0.63) MCL1MEN1KMT2A
SCHEMBL10757133 0.83 ALDH1A1 (0.66) MCL1ALDH1A1CYP1A2POLBKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5760032-A GASTROINTESTINAL DISORDERS AND NERVOUS SYSTEM DISORDERS YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1998-06-02 US disclosed
EP-0776892-A1 THIENYLAZOLE COMPOUND AND THIENOTRIAZOLODIAZEPINE COMPOUND YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1997-06-04 EP disclosed