SCHEMBL8693733

SCHEMBL8693733

CNc1ncccc1C(=O)c1ccccc1

nearest known ligand 0.57

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 5/20 0.57
RAB9A P51151 4/20 0.51
NPC1 O15118 3/20 0.51
HTT P42858 1/20 0.49
KMT2A Q03164 5/20 0.49
AKR1C3 P42330 1/20 0.48
ALDH1A1 P00352 3/20 0.46
GAA P10253 2/20 0.46
MAPT P10636 2/20 0.46
MEN1 O00255 2/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
HPGD P15428 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8696056 0.85 RAB9A (0.52) DHODHRAB9ANPC1KMT2AALDH1A1
SCHEMBL8693815 0.84 DHODH (0.52) DHODHRAB9ANPC1HTTKMT2A
SCHEMBL8696115 0.84 DHODH (0.52) DHODHRAB9ANPC1HTTKMT2A
SCHEMBL29712338 0.84 DHODH (0.64) DHODHRAB9ANPC1HTTKMT2A
SCHEMBL1375514 0.84 DHODH (0.64) DHODHRAB9ANPC1HTTKMT2A
SCHEMBL9842635 0.83 RAB9A (0.68) DHODHRAB9ANPC1HTTKMT2A
SCHEMBL8694084 0.83 DHODH (0.76) DHODHRAB9ANPC1HTTKMT2A
SCHEMBL8691222 0.83 L3MBTL1 (0.54) DHODHRAB9ANPC1HTTKMT2A
SCHEMBL8692652 0.83 POLB (0.55) RAB9ANPC1HTTKMT2AALDH1A1
SCHEMBL13483909 0.83 KMT2A (0.61) DHODHRAB9ANPC1HTTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1043993-C Nonel naphthyridine derivatives and medical composition thereof YAMANOUCHI PHARMA CO LTD (JP) 1999-07-07 CN disclosed
US-5817670-A RESPIRATORY SYSTEM DISORDERS, ORGAN TRANSPLANTATION, ANTITUMOR AGENTS YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1998-10-06 US disclosed
CN-1156455-A Nonel naphthyridine derivatives and medical composition thereof YAMANOUCHI PHARMACUEITCAL CO L (JP) 1997-08-06 CN disclosed
EP-0779292-A1 NOVEL NAPHTHYRIDINE DERIVATIVE AND MEDICINAL COMPOSITION THEREOF YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1997-06-18 EP disclosed