SCHEMBL8694101

SCHEMBL8694101

CNc1ccc(-c2cc(C(F)(F)F)nn2NS(=O)(=O)c2ccccc2)cc1F

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 7/20 0.44
PTGS1 P23219 5/20 0.44
F10 P00742 8/20 0.39
KIF11 P52732 1/20 0.39
PDPK1 O15530 2/20 0.38
F2 P00734 2/20 0.38
KLKB1 P03952 1/20 0.38
PROC P04070 1/20 0.38
PRSS1 P07477 1/20 0.38
RXRA P19793 1/20 0.37
NR1H2 P55055 1/20 0.37
NR1H3 Q13133 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8688899 0.89 PTGS2 (0.44) PTGS2PTGS1PDPK1RXRANR1H2
SCHEMBL8689185 0.88 PTGS2 (0.57) PTGS2PTGS1PDPK1RXRANR1H2
SCHEMBL8688926 0.87 PTGS2 (0.42) PTGS2PTGS1PDPK1RXRANR1H2
SCHEMBL8727373 0.86 PTGS2 (0.48) PTGS2PTGS1PDPK1RXRANR1H2
SCHEMBL8636729 0.85 PTGS2 (0.43) PTGS2PTGS1PDPK1RXRANR1H2
SCHEMBL8652506 0.84 PTGS2 (0.54) PTGS2PTGS1PDPK1RXRANR1H2
SCHEMBL8635943 0.84 PTGS2 (0.41) PTGS2PTGS1PDPK1RXRANR1H2
SCHEMBL8688501 0.84 PTGS2 (0.44) PTGS2PTGS1KIF11PDPK1RXRA
SCHEMBL8640455 0.84 PTGS2 (0.45) PTGS2PTGS1
SCHEMBL8691414 0.84 PTGS2 (0.56) PTGS2PTGS1F10PDPK1RXRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5760068-A NONSTEROIDAL ANTIINFLAMMATORY AGENTS WITH REDUCED SIDE EFFECTS G.D. SEARLE & CO. (US) 1998-06-02 US disclosed
US-5756529-A ANTIINFLAMMATORY G.D. SEARLE & CO. (US) 1998-05-26 US disclosed