SCHEMBL8694124

SCHEMBL8694124

CCCN(CCC)C(=O)Nc1nn(Cc2ccccc2)cc1C(=O)OCC

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.50
LMNA P02545 2/20 0.50
TSHR P16473 1/20 0.43
KDM4E B2RXH2 1/20 0.43
AGTR1 P30556 2/20 0.43
P2RX7 Q99572 1/20 0.42
MAPK1 P28482 2/20 0.41
CREBBP Q92793 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.40
POLB P06746 1/20 0.40
CRHBP P24387 1/20 0.40
CRHR2 Q13324 1/20 0.40
HPGD P15428 1/20 0.40
HTT P42858 1/20 0.39
EGFR P00533 1/20 0.39
ERBB2 P04626 1/20 0.39
CASP3 P42574 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8698593 0.94 ALDH1A1 (0.46) ALDH1A1LMNATSHRKDM4EAGTR1
SCHEMBL8693505 0.91 ALDH1A1 (0.49) ALDH1A1LMNATSHRKDM4EAGTR1
SCHEMBL8696320 0.88 ALDH1A1 (0.50) ALDH1A1LMNATSHRKDM4EAGTR1
SCHEMBL8692534 0.86 AGTR1 (0.49) ALDH1A1LMNATSHRKDM4EAGTR1
SCHEMBL8698769 0.85 ALDH1A1 (0.45) ALDH1A1LMNATSHRKDM4EAGTR1
SCHEMBL8694190 0.85 KDM4E (0.41) ALDH1A1LMNATSHRKDM4ESMN1; SMN2
SCHEMBL8693064 0.84 ALDH1A1 (0.52) ALDH1A1LMNATSHRKDM4EAGTR1
SCHEMBL8693052 0.83 TEAD2 (0.40) TSHRKDM4ESMN1; SMN2POLBHPGD
SCHEMBL8593357 0.82 ALDH1A1 (0.48) ALDH1A1LMNATSHRKDM4EAGTR1
SCHEMBL8696794 0.82 ALDH1A1 (0.48) ALDH1A1LMNATSHRKDM4EAGTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5849779-A Pyrazole derivatives and their pharmaceutical use JAPAN ENERGY CORPORATION (JP) 1998-12-15 US disclosed
EP-0810217-A1 Pyrazole derivatives and their pharmaceutical use as smooth muscle cell growth inhibitors JAPAN ENERGY CORPORATION (JP) 1997-12-03 EP disclosed