SCHEMBL8698769

SCHEMBL8698769

CCCCN(CCCC)C(=S)Nc1nn(Cc2ccccc2)cc1C(=O)OCC

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.45
LMNA P02545 3/20 0.45
AGTR1 P30556 2/20 0.41
KDM4E B2RXH2 1/20 0.41
CREBBP Q92793 1/20 0.41
TSHR P16473 1/20 0.41
P2RX7 Q99572 1/20 0.40
MAPK1 P28482 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
POLB P06746 1/20 0.39
CRHBP P24387 1/20 0.38
CRHR2 Q13324 1/20 0.38
EGFR P00533 2/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
RXFP1 Q9HBX9 1/20 0.37
FOS P01100 1/20 0.37
JUN P05412 1/20 0.37
NFKB1 P19838 1/20 0.37
NFKB2 Q00653 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8693505 0.94 ALDH1A1 (0.49) ALDH1A1LMNAAGTR1KDM4ECREBBP
SCHEMBL8698593 0.91 ALDH1A1 (0.46) ALDH1A1LMNAAGTR1KDM4ECREBBP
SCHEMBL8696794 0.88 ALDH1A1 (0.48) ALDH1A1LMNAAGTR1KDM4ECREBBP
SCHEMBL8693996 0.86 AGTR1 (0.47) ALDH1A1LMNAAGTR1KDM4ECREBBP
SCHEMBL8696980 0.86 TEAD2 (0.37) ALDH1A1LMNAKDM4ESMN1; SMN2FOS
SCHEMBL8692506 0.86 TEAD2 (0.39) ALDH1A1LMNAKDM4ETSHRSMN1; SMN2
SCHEMBL8694124 0.85 ALDH1A1 (0.50) ALDH1A1LMNAAGTR1KDM4ECREBBP
SCHEMBL8694236 0.84 ALDH1A1 (0.46) ALDH1A1LMNAAGTR1KDM4ECREBBP
SCHEMBL8693140 0.83 ALDH1A1 (0.45) ALDH1A1LMNAAGTR1KDM4ECREBBP
SCHEMBL8696343 0.82 ALDH1A1 (0.47) ALDH1A1LMNAAGTR1KDM4ECREBBP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5849779-A Pyrazole derivatives and their pharmaceutical use JAPAN ENERGY CORPORATION (JP) 1998-12-15 US disclosed
EP-0810217-A1 Pyrazole derivatives and their pharmaceutical use as smooth muscle cell growth inhibitors JAPAN ENERGY CORPORATION (JP) 1997-12-03 EP disclosed