SCHEMBL8696129

SCHEMBL8696129

CCOC(=O)c1cn(C2CC2)c2c(Cl)c(Cl)nc(C)c2c1=O

nearest known ligand 0.56

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 1/20 0.44
STAT3 P40763 1/20 0.42
TOP2A P11388 4/20 0.39
TOP2B Q02880 4/20 0.39
TDP1 Q9NUW8 1/20 0.38
TSHR P16473 1/20 0.38
CASP1 P29466 1/20 0.38
POLB P06746 2/20 0.37
HTT P42858 2/20 0.37
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
CYP1A2 P05177 1/20 0.37
KMT2A Q03164 1/20 0.37
BAZ2B Q9UIF8 1/20 0.37
BAZ2A Q9UIF9 1/20 0.37
KDM5B Q9UGL1 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7840898 0.85 TOP2A (0.52) TOP2ATOP2BPOLBKDM4EALDH1A1
SCHEMBL7842470 0.83 ADRB2 (0.34) ADRB2TOP2ATOP2BPOLBALDH1A1
SCHEMBL8692136 0.83 ADRB2 (0.47) ADRB2STAT3TOP2ATOP2BTDP1
SCHEMBL9133982 0.82 ADRB2 (0.50) ADRB2STAT3TOP2ATOP2BTSHR
SCHEMBL8116592 0.80 ADRB2 (0.49) ADRB2STAT3TOP2ATOP2BTSHR
SCHEMBL9585893 0.79 STAT3 (0.54) ADRB2STAT3TOP2ATOP2BTSHR
SCHEMBL5704330 0.79 ADRB2 (0.49) ADRB2STAT3TOP2ATOP2BTSHR
SCHEMBL9688633 0.79 CACNA1F (0.49) ADRB2STAT3TOP2ATOP2BPOLB
SCHEMBL8696955 0.79 STAT3 (0.43) STAT3TDP1TSHRCASP1POLB
SCHEMBL7840900 0.78 TOP2A (0.37) TOP2ATOP2BPOLBALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5811433-A ANTIMICROBIALS BAYER AKTIENGESELLSCHAFT (DE) 1998-09-22 US disclosed