SCHEMBL7842470

SCHEMBL7842470

CCOC(=O)Oc1cn(C2CC2)c2c(Cl)c(Cl)nc(C)c2c1=O

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 1/20 0.34
TOP2A P11388 6/20 0.33
TOP2B Q02880 6/20 0.33
TNF P01375 1/20 0.33
KCNH2 Q12809 2/20 0.33
CUL4A Q13619 1/20 0.32
TYMS P04818 1/20 0.32
MAPT P10636 1/20 0.30
ALDH1A1 P00352 1/20 0.30
POLB P06746 1/20 0.30
CHRM2 P08172 1/20 0.30
CHRM1 P11229 1/20 0.30
OPRM1 P35372 1/20 0.30
OPRD1 P41143 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7840900 0.87 TOP2A (0.37) TOP2ATOP2BKCNH2ALDH1A1POLB
SCHEMBL7850179 0.87 CYP3A4 (0.31) CUL4ATYMS
SCHEMBL7840741 0.83 ADRB2 (0.34) ADRB2TOP2ATOP2BTNFKCNH2
SCHEMBL8696129 0.83 ADRB2 (0.44) ADRB2TOP2ATOP2BALDH1A1POLB
SCHEMBL7503528 0.78 ADRB2 (0.40) ADRB2TOP2ATOP2BKCNH2
SCHEMBL9687476 0.77 CUL4A (0.36) ADRB2TOP2ATOP2BTNFCUL4A
SCHEMBL7840898 0.77 TOP2A (0.52) TOP2ATOP2BKCNH2ALDH1A1POLB
SCHEMBL7817401 0.76 ADRB2 (0.47) ADRB2TOP2ATOP2BKCNH2ALDH1A1
SCHEMBL9416462 0.76 TNF (0.35) TNFMAPTALDH1A1POLB
SCHEMBL7095727 0.76 DPP4 (0.40) ADRB2TOP2ATOP2BKCNH2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726270-B1 Derivatives of 1,6-naphthyridone carboxylic acids BAYER AG (DE) 2001-05-23 EP disclosed
EP-0726270-A1 Derivatives of 1,6-naphthyridine carboxylic acids BAYER AG (DE) 1996-08-14 EP disclosed