SCHEMBL8696141

SCHEMBL8696141

CCC(c1ccccc1)N(C(=O)OC(C)(C)C)c1c(-c2cc(C)cc(C)c2)[nH]c2ccc(N)cc12

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGES O14684 1/20 0.34
ALOX5 P09917 1/20 0.34
GABRA1 P14867 3/20 0.34
GABRG2 P18507 3/20 0.34
GABRB3 P28472 3/20 0.34
GABRA5 P31644 3/20 0.34
GABRA3 P34903 3/20 0.34
GABRA2 P47869 3/20 0.34
ALDH1A1 P00352 3/20 0.34
MAPT P10636 3/20 0.34
GABRA6 Q16445 2/20 0.34
KDM4E B2RXH2 2/20 0.34
GAA P10253 2/20 0.34
HPGD P15428 2/20 0.34
HSD17B10 Q99714 2/20 0.34
MEN1 O00255 1/20 0.34
LMNA P02545 1/20 0.34
MAPK10 P53779 1/20 0.34
KMT2A Q03164 1/20 0.34
CACNA1B Q00975 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8696137 0.79 MEN1 (0.38) PTGESALOX5ALDH1A1MAPTKDM4E
SCHEMBL6983626 0.73 HDAC1 (0.48) HDAC1
SCHEMBL7970722 0.65 TRPM8 (0.42) ALOX5LMNAHDAC1TRPM8
SCHEMBL17776389 0.65 CHRNB2 (0.44) KDM4EGAAHDAC1TRPM8
SCHEMBL3051043 0.62 ADRB2 (0.37) ALDH1A1KDM4ETP53SMN1; SMN2
SCHEMBL29913609 0.60 TRPM8 (0.39) ALDH1A1GAALMNAHDAC1SMN1; SMN2
SCHEMBL7636101 0.60 KDM4E (0.49) GABRA1GABRG2GABRB3GABRA3GABRA2
SCHEMBL23609358 0.60 S1PR3 (0.32) KMT2AGABRB1GABRB2
SCHEMBL7408450 0.60 GAA (0.44) KDM4EGAA
SCHEMBL31016664 0.60 GAA (0.44) KDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5780437-A ADMINISTERING TO TREAT SEX-HORMONE RELATED DISORDERS MERCK & CO., INC. (US) 1998-07-14 US disclosed