SCHEMBL8696809

SCHEMBL8696809

CCOC(=O)c1cnn(-c2ccccc2)c1NC(=S)Nc1ccccc1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 10/20 0.71
RAB9A P51151 5/20 0.67
HTT P42858 3/20 0.67
NPSR1 Q6W5P4 4/20 0.63
KDM4E B2RXH2 1/20 0.63
HPGD P15428 3/20 0.59
NPC1 O15118 4/20 0.58
GAA P10253 1/20 0.58
L3MBTL1 Q9Y468 1/20 0.58
LMNA P02545 1/20 0.56
SMN1; SMN2 Q16637 4/20 0.56
MAPT P10636 2/20 0.54
MEN1 O00255 1/20 0.54
ALOX12 P18054 1/20 0.54
KMT2A Q03164 1/20 0.54
GPR35 Q9HC97 1/20 0.53
GPR55 Q9Y2T6 1/20 0.53
NFKB1 P19838 1/20 0.51
NFKB2 Q00653 1/20 0.51
RELA Q04206 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8699832 0.89 ALDH1A1 (0.73) ALDH1A1RAB9AHTTNPSR1KDM4E
SCHEMBL8693125 0.87 ALDH1A1 (0.70) ALDH1A1RAB9AHTTNPSR1KDM4E
SCHEMBL13975009 0.84 ALDH1A1 (0.77) ALDH1A1RAB9AHTTNPSR1KDM4E
SCHEMBL8696906 0.83 NPC1 (0.59) ALDH1A1RAB9AHTTNPSR1KDM4E
SCHEMBL3516960 0.82 ALDH1A1 (0.74) ALDH1A1RAB9AHTTNPSR1KDM4E
SCHEMBL7934013 0.82 ALDH1A1 (0.79) ALDH1A1RAB9AHTTNPSR1KDM4E
SCHEMBL4158508 0.82 ALDH1A1 (0.79) ALDH1A1RAB9AHTTNPSR1KDM4E
SCHEMBL9010473 0.82 ALDH1A1 (0.79) ALDH1A1RAB9AHTTNPSR1KDM4E
SCHEMBL8696284 0.80 ALDH1A1 (0.72) ALDH1A1RAB9AHTTNPSR1KDM4E
SCHEMBL13235027 0.79 ALDH1A1 (0.65) ALDH1A1RAB9AHTTNPSR1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5849779-A Pyrazole derivatives and their pharmaceutical use JAPAN ENERGY CORPORATION (JP) 1998-12-15 US disclosed
EP-0810217-A1 Pyrazole derivatives and their pharmaceutical use as smooth muscle cell growth inhibitors JAPAN ENERGY CORPORATION (JP) 1997-12-03 EP disclosed