SCHEMBL8697131

SCHEMBL8697131

NS(=O)(=O)c1ccccc1-c1ccccc1-c1ncccn1

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CA1 P00915 6/20 0.47
CA2 P00918 6/20 0.47
CA9 Q16790 4/20 0.47
MAPK1 P28482 1/20 0.47
ALOX5AP P20292 4/20 0.46
FEN1 P39748 4/20 0.46
CA6 P23280 3/20 0.44
CA4 P22748 2/20 0.44
CA12 O43570 2/20 0.44
CA5A P35218 2/20 0.44
CA7 P43166 2/20 0.44
CA5B Q9Y2D0 2/20 0.44
CYP2C9 P11712 1/20 0.44
CA14 Q9ULX7 1/20 0.44
EDNRA P25101 1/20 0.41
FTO Q9C0B1 1/20 0.40
LMNA P02545 1/20 0.40
PTPRC P08575 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1094361 0.92 CA1 (0.50) CA1CA2CA9MAPK1ALOX5AP
Pyrimidine SCHEMBL16180729 0.84 CA1 (0.44) CA1CA2CA9MAPK1ALOX5AP
SCHEMBL8347239 0.84 CA2 (0.58) CA1CA2CA9MAPK1ALOX5AP
SCHEMBL8697589 0.82 ALOX5AP (0.47) CA1CA2CA9MAPK1ALOX5AP
SCHEMBL1080972 0.82 CA2 (0.61) CA1CA2CA9ALOX5APFEN1
SCHEMBL7974328 0.80 CA1 (0.46) CA1CA2CA9MAPK1ALOX5AP
SCHEMBL1667127 0.78 EDNRA (0.49) CA1CA2CA9MAPK1ALOX5AP
SCHEMBL29967288 0.78 EDNRA (0.49) CA1CA2CA9MAPK1ALOX5AP
SCHEMBL12853990 0.77 PTPRC (0.44) LMNAPTPRC
SCHEMBL3256397 0.76 CA1 (0.73) CA1CA2CA9MAPK1CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998004260-A1 SUBSTITUTED BIPHENYL SULFONAMIDE ENDOTHELIN ANTAGONISTS BRISTOL-MYERS SQUIBB COMPANY (US) 1998-02-05 WO claimed