SCHEMBL7974328

SCHEMBL7974328

NS(=O)(=O)c1ccccc1-c1ccnc(-c2ncccn2)n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 5/20 0.46
CA2 P00918 5/20 0.46
CA9 Q16790 3/20 0.46
MAPK1 P28482 1/20 0.46
ALOX5AP P20292 5/20 0.45
FEN1 P39748 5/20 0.45
CA4 P22748 2/20 0.39
CA6 P23280 2/20 0.39
IKBKB O14920 1/20 0.39
CA12 O43570 1/20 0.39
CYP2C9 P11712 1/20 0.39
CA5A P35218 1/20 0.39
CA7 P43166 1/20 0.39
CA14 Q9ULX7 1/20 0.39
CA5B Q9Y2D0 1/20 0.39
F2 P00734 1/20 0.36
F10 P00742 1/20 0.36
PRSS1 P07477 1/20 0.36
PRSS2 P07478 1/20 0.36
PRSS3 P35030 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1094361 0.83 CA1 (0.50) CA1CA2CA9MAPK1ALOX5AP
SCHEMBL29967288 0.80 EDNRA (0.49) CA1CA2CA9MAPK1ALOX5AP
SCHEMBL1667127 0.80 EDNRA (0.49) CA1CA2CA9MAPK1ALOX5AP
SCHEMBL8697131 0.80 CA1 (0.47) CA1CA2CA9MAPK1ALOX5AP
SCHEMBL30372027 0.76 TGFBR1 (0.42) CA1CA2CA9MAPK1ALOX5AP
Pyrimidine SCHEMBL16180729 0.75 CA1 (0.44) CA1CA2CA9MAPK1ALOX5AP
SCHEMBL1094172 0.75 CA2 (0.44) CA1CA2CA9MAPK1ALOX5AP
SCHEMBL8697589 0.73 ALOX5AP (0.47) CA1CA2CA9MAPK1ALOX5AP
SCHEMBL7868583 0.73 CDK9 (0.40) CA1CA2CA9ALOX5APFEN1
SCHEMBL4669011 0.72 ALOX5AP (0.49) CA1CA2CA9MAPK1ALOX5AP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001081335-A1 PYRIMIDINE-SULFONAMIDES HAVING ENDOTHELIN-ANTAGONIST ACTIVITY ACTELION PHARMACEUTICALS LTD (CH) 2001-11-01 WO claimed