SCHEMBL8697744

SCHEMBL8697744

CCCCCC(N[C]=O)c1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 3/20 0.42
NAAA Q02083 2/20 0.41
POLB P06746 1/20 0.41
CNR2 P34972 1/20 0.41
ASAH1 Q13510 2/20 0.39
SLC2A1 P11166 1/20 0.39
ALDH1A1 P00352 1/20 0.38
ACER2 Q5QJU3 1/20 0.38
GPR88 Q9GZN0 1/20 0.38
SIGMAR1 Q99720 1/20 0.38
NPC1 O15118 1/20 0.38
LMNA P02545 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
MMP2 P08253 2/20 0.37
MMP9 P14780 2/20 0.37
MMP1 P03956 1/20 0.37
MMP3 P08254 1/20 0.37
MMP14 P50281 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8701351 0.95 POLB (0.45) TACR3NAAAPOLBCNR2ASAH1
SCHEMBL3368388 0.88 AOC3 (0.42) TACR3POLBALDH1A1GPR88LMNA
SCHEMBL5640387 0.80 LMNA (0.46) POLBALDH1A1NPC1LMNA
SCHEMBL14533565 0.79 ALDH1A1 (0.45) TACR3NAAAPOLBCNR2SLC2A1
SCHEMBL7754951 0.77 TACR3 (0.44) TACR3NAAAPOLBCNR2ASAH1
SCHEMBL11256309 0.77 TACR3 (0.44) TACR3NAAAASAH1SLC2A1ALDH1A1
SCHEMBL27462652 0.77 SLC2A1 (0.55) TACR3NAAAPOLBCNR2ASAH1
SCHEMBL10356497 0.77 TACR3 (0.44) TACR3NAAAPOLBCNR2ASAH1
SCHEMBL11153215 0.77 TACR3 (0.44) TACR3NAAAASAH1SLC2A1ALDH1A1
SCHEMBL9149427 0.77 TACR3 (0.44) TACR3NAAAASAH1SLC2A1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5834460-A FOR TREATMENT OF BRAIN OR PSYCHOLOGICAL DISORDERS, ALZHEIMER*S DISEASE, MENTAL RETARDATION OR AUTISM YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1998-11-10 US disclosed
EP-0696586-A1 SERINE DERIVATIVE YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1996-02-14 EP disclosed
EP-0377633-B1 PEROXIDE FREE RADICAL INITIATORS CONTAINING HINDERED AMINE LIGHT STABILIZER GROUPS ATOCHEM NORTH AMERICA (US) 1995-05-17 EP disclosed
EP-0377633-A4 PEROXIDE FREE RADICAL INITIATORS CONTAINING HINDERED AMINE LIGHT STABILIZER GROUPS 1991-01-30 EP disclosed
EP-0377633-A1 PEROXIDE FREE RADICAL INITIATORS CONTAINING HINDERED AMINE LIGHT STABILIZER GROUPS. PENNWALT CORP (US) 1990-07-18 EP disclosed
US-4925903-A PEROXIDE CONTAINING HINDERED AMINE ALSO FUNCTIONS AS INITIATOR PENNWALT CORPORATION (US) 1990-05-15 US disclosed
US-4885347-A UNSATURATED POLYESTER PENNWALT CORPORATION (US) 1989-12-05 US disclosed
WO-1989001474-A1 PEROXIDE FREE RADICAL INITIATORS CONTAINING HINDERED AMINE LIGHT STABILIZER GROUPS PENNWALT CORPORATION (US) 1989-02-23 WO disclosed
EP-0294818-A2 Hindered amine light stabilizers containing aromatic carboxy groups and derivatives ELF ATOCHEM NORTH AMERICA, INC. (US) 1988-12-14 EP disclosed