SCHEMBL8697882

SCHEMBL8697882

Cc1ccc(C(F)(c2cncnc2)c2ccc(-c3ccccc3)o2)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 6/20 0.40
NPC1 O15118 5/20 0.35
RAB9A P51151 5/20 0.35
HPGD P15428 4/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
POLB P06746 1/20 0.35
NFKB1 P19838 1/20 0.35
NFKB2 Q00653 1/20 0.35
RELA Q04206 1/20 0.35
CASP3 P42574 1/20 0.34
SENP8 Q96LD8 1/20 0.34
SENP7 Q9BQF6 1/20 0.34
SENP6 Q9GZR1 1/20 0.34
KMT2A Q03164 3/20 0.34
GAA P10253 2/20 0.34
KDM4E B2RXH2 3/20 0.33
ALDH1A1 P00352 3/20 0.33
MEN1 O00255 2/20 0.33
HSD17B10 Q99714 2/20 0.33
ATM Q13315 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8702192 0.91 CYP19A1 (0.41) CYP19A1NPC1RAB9AHPGDKMT2A
SCHEMBL8697579 0.88 CYP19A1 (0.51) CYP19A1NPC1RAB9AHPGDPOLB
SCHEMBL8699069 0.87 CYP19A1 (0.57) CYP19A1NPC1RAB9A
SCHEMBL8698474 0.84 CYP19A1 (0.38) CYP19A1NPC1RAB9A
SCHEMBL8697545 0.82 CYP19A1 (0.57) CYP19A1NPC1RAB9AHPGDSMN1; SMN2
SCHEMBL8698611 0.77 CYP19A1 (0.41) CYP19A1ATMMAOB
SCHEMBL8697385 0.74 CYP19A1 (0.46) CYP19A1NPC1RAB9AHPGDSMN1; SMN2
SCHEMBL8702199 0.74 CYP19A1 (0.45) CYP19A1NPC1RAB9ASMN1; SMN2POLB
SCHEMBL8697944 0.72 CYP3A4 (0.43) CYP19A1TSHR
SCHEMBL8702833 0.72 CYP19A1 (0.57) CYP19A1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998018791-A1 HETEROCYCLIC FURAN COMPOUNDS, THEIR PREPARATION AND USE AS AROMATASE INHIBITORS A. MENARINI INDUSTRIE FARMACEUTICHE RIUNITE S.R.L. (IT) 1998-05-07 WO claimed
WO-1998018791-A1 HETEROCYCLIC FURAN COMPOUNDS, THEIR PREPARATION AND USE AS AROMATASE INHIBITORS A. MENARINI INDUSTRIE FARMACEUTICHE RIUNITE S.R.L. (IT) 1998-05-07 WO disclosed