SCHEMBL8702192

SCHEMBL8702192

FC(c1ccccc1)(c1cncnc1)c1ccc(-c2ccccc2)o1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 7/20 0.41
ATM Q13315 1/20 0.38
ALOX15 P16050 1/20 0.36
TSHR P16473 1/20 0.36
CASP1 P29466 1/20 0.36
RAB9A P51151 3/20 0.35
KDM4E B2RXH2 1/20 0.35
NPC1 O15118 1/20 0.35
ALDH1A1 P00352 1/20 0.35
HPGD P15428 1/20 0.35
HSD17B10 Q99714 1/20 0.35
NOTUM Q6P988 1/20 0.33
CCNC P24863 1/20 0.33
CDK8 P49336 1/20 0.33
PDE4B Q07343 1/20 0.33
CYP2E1 P05181 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2A6 P11509 1/20 0.33
CYP2C9 P11712 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8697579 0.92 CYP19A1 (0.51) CYP19A1ATMALOX15TSHRCASP1
SCHEMBL8699069 0.91 CYP19A1 (0.57) CYP19A1RAB9ANPC1CYP3A4
SCHEMBL8697882 0.91 CYP19A1 (0.40) CYP19A1ATMALOX15TSHRCASP1
SCHEMBL8698474 0.87 CYP19A1 (0.38) CYP19A1RAB9ANPC1CYP3A4
SCHEMBL8698611 0.82 CYP19A1 (0.41) CYP19A1ATMCCNCCDK8CYP3A4
SCHEMBL8698102 0.79 CYP19A1 (0.51) CYP19A1ATMALOX15TSHRCASP1
SCHEMBL8697944 0.78 CYP3A4 (0.43) CYP19A1TSHRCYP3A4CYP2D6CYP2C19
SCHEMBL8700748 0.77 CYP3A4 (0.36) CYP19A1TSHRCYP3A4CYP2D6CYP2C19
SCHEMBL8702833 0.74 CYP19A1 (0.57) CYP19A1RAB9ACYP3A4
SCHEMBL8700104 0.74 CYP19A1 (0.45) CYP19A1ATMTSHRKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998018791-A1 HETEROCYCLIC FURAN COMPOUNDS, THEIR PREPARATION AND USE AS AROMATASE INHIBITORS A. MENARINI INDUSTRIE FARMACEUTICHE RIUNITE S.R.L. (IT) 1998-05-07 WO disclosed