SCHEMBL8698706

SCHEMBL8698706

CCCCn1cc(C(=O)O)c(NC(=S)NCCC)n1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 1/20 0.46
KMT2A Q03164 1/20 0.40
GAA P10253 4/20 0.39
KDM4E B2RXH2 3/20 0.39
MAPT P10636 2/20 0.36
ALOX12 P18054 2/20 0.36
ALDH1A1 P00352 5/20 0.36
CYP1A2 P05177 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
SMN1; SMN2 Q16637 3/20 0.35
HPGD P15428 1/20 0.35
QPCT Q16769 1/20 0.34
ALPL P05186 1/20 0.34
SIGMAR1 Q99720 1/20 0.34
LMNA P02545 2/20 0.34
KDM4C Q9H3R0 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8693969 0.95 HCAR2 (0.46) HCAR2KMT2AGAAKDM4EMAPT
SCHEMBL8696838 0.93 HCAR2 (0.44) HCAR2GAAKDM4EALDH1A1SMN1; SMN2
SCHEMBL8694003 0.93 KMT2A (0.41) HCAR2KMT2AGAAKDM4EMAPT
SCHEMBL8698707 0.90 GAA (0.44) HCAR2KMT2AGAAKDM4EMAPT
SCHEMBL8693702 0.89 KMT2A (0.42) HCAR2KMT2AGAAKDM4EMAPT
SCHEMBL8693069 0.88 KDM4E (0.41) HCAR2GAAKDM4EALDH1A1SMN1; SMN2
SCHEMBL8693503 0.88 HCAR2 (0.47) HCAR2KMT2AKDM4EALDH1A1CYP1A2
SCHEMBL8693176 0.86 GAA (0.42) HCAR2KMT2AGAAKDM4EMAPT
SCHEMBL8693750 0.86 ALDH1A1 (0.41) HCAR2KMT2AGAAKDM4EMAPT
SCHEMBL8694654 0.84 KDM4E (0.39) HCAR2GAAKDM4EALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5849779-A Pyrazole derivatives and their pharmaceutical use JAPAN ENERGY CORPORATION (JP) 1998-12-15 US disclosed
EP-0810217-A1 Pyrazole derivatives and their pharmaceutical use as smooth muscle cell growth inhibitors JAPAN ENERGY CORPORATION (JP) 1997-12-03 EP disclosed