SCHEMBL8699425

SCHEMBL8699425

O=C(O)C1=CC2=Cc3ccccc3C2=N1

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 1/20 0.40
MAOA P21397 1/20 0.33
MAOB P27338 1/20 0.33
CA12 O43570 2/20 0.31
CA9 Q16790 2/20 0.31
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31
SCN2A Q99250 1/20 0.31
LMNA P02545 1/20 0.31
ALOX15 P16050 2/20 0.30
DAO P14920 1/20 0.30
TSHR P16473 1/20 0.30
NAPRT Q6XQN6 1/20 0.30
ALDH1A1 P00352 1/20 0.30
POLB P06746 1/20 0.30
KMT2A Q03164 1/20 0.30
MAPT P10636 1/20 0.30
HTT P42858 1/20 0.30
HBB P68871 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30895284 0.69 MAOA (0.50) MAOAMAOBCA12CA9CA1
SCHEMBL503745 0.69 MAOA (0.50) MAOAMAOBCA12CA9CA1
Hydrochloric Acid SCHEMBL26614007 0.67 MAOA (0.48) MAOAMAOBCA12CA9CA1
Ethylene SCHEMBL28442445 0.66 MAOA (0.47) MAOAMAOBCA12CA9CA1
SCHEMBL7354968 0.64 MAOA (0.50) MAOAMAOBCA12CA9CA1
SCHEMBL8155087 0.64
Ethylene Glycol SCHEMBL8419054 0.63 MAOA (0.49) MAOAMAOBCA12CA9CA1
SCHEMBL28211937 0.63 MAOA (0.49) MAOAMAOBCA12CA9CA1
SCHEMBL30493712 0.61 ABCG2 (0.38) ABCG2
SCHEMBL1864060 0.61 ABCG2 (0.38) ABCG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998042709-A1 ENDOTHELIN-RECEPTOR ANTAGONISTS MERCK PATENT GMBH (DE) 1998-10-01 WO disclosed