SCHEMBL8699650

SCHEMBL8699650

O=C1CC(=O)c2ccncc2C1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.39
MAOB P27338 1/20 0.39
CDC25B P30305 1/20 0.38
PDE3B Q13370 2/20 0.38
PDE3A Q14432 2/20 0.38
CYP1A2 P05177 3/20 0.38
SIGMAR1 Q99720 1/20 0.38
CYP11B1 P15538 2/20 0.36
CYP11B2 P19099 2/20 0.36
CYP3A4 P08684 3/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
CHRNB2 P17787 1/20 0.34
CHRNA4 P43681 1/20 0.34
CYP19A1 P11511 3/20 0.34
NPSR1 Q6W5P4 1/20 0.33
TP53 P04637 2/20 0.32
MAPT P10636 2/20 0.32
CASP1 P29466 2/20 0.32
BLM P54132 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7343370 0.79 CYP1A2 (0.50) MAOAMAOBCDC25BPDE3BPDE3A
SCHEMBL29699898 0.75 SIGMAR1 (0.48) MAOAMAOBCDC25BPDE3BPDE3A
SCHEMBL14452876 0.75 SIGMAR1 (0.48) MAOAMAOBCDC25BPDE3BPDE3A
SCHEMBL4323285 0.75 CYP1A2 (0.53) MAOAMAOBCDC25BPDE3BPDE3A
SCHEMBL29792666 0.75 CYP1A2 (0.53) MAOAMAOBCDC25BPDE3BPDE3A
SCHEMBL20718539 0.74 MAOA (0.50) MAOAMAOBCDC25BPDE3BPDE3A
SCHEMBL11265174 0.72 SIGMAR1 (0.57) MAOAMAOBCDC25BPDE3BPDE3A
SCHEMBL2877256 0.72 MAOA (0.53) MAOAMAOBCDC25BCYP1A2SIGMAR1
SCHEMBL31128508 0.72 MAOA (0.53) MAOAMAOBCDC25BCYP1A2SIGMAR1
SCHEMBL8936257 0.71 SIGMAR1 (0.32) MAOAMAOBCYP1A2SIGMAR1CYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108640914-B Method for synthesizing isoindole [2,1-b ] isoquinoline-5, 7-diketone compound 河南师范大学 2020-07-31 CN claimed
CN-108467393-B Method for synthesizing isoindole [2,1-b ] isoquinoline-5, 7-diketone compounds by three components in one pot 河南师范大学 2020-06-02 CN claimed
CN-108467393-A The method of one pot of three component synthesis iso-indoles [2,1-b] isoquinolin -5,7- cyclohexadione compounds 河南师范大学 2018-08-31 CN disclosed
US-5733918-A ANTITUMOR AGENT TAIHO PHARMACEUTICAL CO., LTD. (JP) 1998-03-31 US disclosed
US-5710162-A ANTITUMOR AGENTS TAIHO PHARMACEUTICAL CO., LTD. (JP) 1998-01-20 US disclosed