SCHEMBL8700449

SCHEMBL8700449

CCOC(=O)Oc1c(-c2ccc(OC)cc2)c2c(c3ccccc3n2C)n1Cc1ccccc1OC

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
EDNRB P24530 10/20 0.49
KDM4E B2RXH2 5/20 0.44
ALDH1A1 P00352 5/20 0.44
HPGD P15428 5/20 0.44
TSHR P16473 2/20 0.44
KMT2A Q03164 2/20 0.44
USP2 O75604 2/20 0.44
HSD17B10 Q99714 1/20 0.44
KLK7 P49862 1/20 0.44
TP53 P04637 3/20 0.42
SMN1; SMN2 Q16637 1/20 0.41
GNRHR P30968 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6658792 0.89 EDNRB (0.51) EDNRBKDM4EALDH1A1HPGDTSHR
SCHEMBL6659388 0.83 EDNRB (0.53) EDNRBKDM4EALDH1A1HPGDTSHR
SCHEMBL6315607 0.82 EDNRB (0.54) EDNRBKDM4EALDH1A1HPGDTSHR
SCHEMBL8703164 0.78 EDNRB (0.63) EDNRB
SCHEMBL6313381 0.77 EDNRB (0.55) EDNRBKDM4EALDH1A1HPGDTSHR
SCHEMBL8700801 0.77 EDNRB (0.68) EDNRB
SCHEMBL8696580 0.74 ALDH1A1 (0.46) KDM4EALDH1A1HPGDTSHRKMT2A
SCHEMBL8698304 0.70 EDNRB (0.75) EDNRB
SCHEMBL8552678 0.67 EDNRB (0.43) EDNRB
SCHEMBL8552610 0.66 EDNRB (0.46) EDNRBKDM4EALDH1A1KMT2AHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998042709-A1 ENDOTHELIN-RECEPTOR ANTAGONISTS MERCK PATENT GMBH (DE) 1998-10-01 WO disclosed