SCHEMBL8700748

SCHEMBL8700748

N#Cc1ccc(C(F)(c2cncnc2)c2ccc(-c3ccccc3)o2)c(C#N)c1

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.36
CYP3A5 P20815 1/20 0.36
FLT1 P17948 2/20 0.34
FLT4 P35916 2/20 0.34
KDR P35968 2/20 0.34
MAPKAPK2 P49137 2/20 0.31
CYP11B1 P15538 3/20 0.31
CYP11B2 P19099 3/20 0.31
KIF11 P52732 1/20 0.31
CYP19A1 P11511 1/20 0.31
CYP1A2 P05177 1/20 0.30
CYP2D6 P10635 1/20 0.30
TSHR P16473 1/20 0.30
CYP2C19 P33261 1/20 0.30
FNTA P49354 1/20 0.30
FNTB P49356 1/20 0.30
GRM5 P41594 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8697944 0.91 CYP3A4 (0.43) CYP3A4CYP3A5FLT1FLT4KDR
SCHEMBL8698526 0.85 CYP3A4 (0.38) CYP3A4CYP3A5FLT1FLT4KDR
SCHEMBL8698474 0.85 CYP19A1 (0.38) CYP3A4CYP3A5MAPKAPK2CYP11B2KIF11
SCHEMBL8698505 0.80 CYP19A1 (0.38) CYP3A4CYP3A5CYP19A1TSHR
SCHEMBL8697496 0.79 AR (0.41) CYP3A4CYP3A5CYP11B1CYP11B2CYP19A1
SCHEMBL8697489 0.79 CYP3A4 (0.49) CYP3A4CYP3A5FLT1FLT4KDR
SCHEMBL8698611 0.78 CYP19A1 (0.41) CYP3A4CYP11B1CYP11B2CYP19A1
SCHEMBL8702192 0.77 CYP19A1 (0.41) CYP3A4CYP19A1CYP2D6TSHRCYP2C19
SCHEMBL8700497 0.73 CYP19A1 (0.43) CYP3A4CYP3A5CYP11B2CYP19A1FNTA
SCHEMBL8697579 0.73 CYP19A1 (0.51) MAPKAPK2CYP19A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998018791-A1 HETEROCYCLIC FURAN COMPOUNDS, THEIR PREPARATION AND USE AS AROMATASE INHIBITORS A. MENARINI INDUSTRIE FARMACEUTICHE RIUNITE S.R.L. (IT) 1998-05-07 WO claimed
WO-1998018791-A1 HETEROCYCLIC FURAN COMPOUNDS, THEIR PREPARATION AND USE AS AROMATASE INHIBITORS A. MENARINI INDUSTRIE FARMACEUTICHE RIUNITE S.R.L. (IT) 1998-05-07 WO disclosed