SCHEMBL8700922

SCHEMBL8700922

COc1ccc(-c2cc(-c3cccc(C(=O)Cl)n3)nc(-c3cccc(C(=O)Cl)n3)c2)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 5/20 0.53
ADORA3 P0DMS8 1/20 0.47
KDM4E B2RXH2 1/20 0.46
MEN1 O00255 1/20 0.46
GAA P10253 1/20 0.46
KMT2A Q03164 1/20 0.46
CTSA P10619 2/20 0.42
ABL1 P00519 1/20 0.42
ABCB1 P08183 1/20 0.42
BCR P11274 1/20 0.42
FYN P06241 1/20 0.42
LTB4R Q15722 1/20 0.41
CHEK1 O14757 1/20 0.41
PARP1 P09874 2/20 0.41
NPC1 O15118 1/20 0.41
TP53 P04637 1/20 0.41
MAPK1 P28482 1/20 0.41
CASP3 P42574 1/20 0.41
RAB9A P51151 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7772127 0.92 MCL1 (0.49) MCL1ADORA3KDM4EMEN1KMT2A
SCHEMBL8700788 0.88 MCL1 (0.64) MCL1ADORA3LTB4RCHEK1SMN1; SMN2
SCHEMBL14496264 0.85 MCL1 (0.72) MCL1ADORA3
SCHEMBL7770325 0.80 MCL1 (0.59) MCL1ADORA3KDM4EMEN1KMT2A
SCHEMBL7850867 0.76 ABL1 (0.47) MCL1ADORA3KDM4EKMT2AABL1
SCHEMBL8600130 0.75 TERT (0.47) MCL1ADORA3KDM4EKMT2AABL1
SCHEMBL8596986 0.75 ABL1 (0.44) MCL1ADORA3KDM4EABL1ABCB1
SCHEMBL14008675 0.75 FAAH (0.52) MCL1KDM4EGAASMN1; SMN2
SCHEMBL4630405 0.74 MCL1 (0.60) MCL1ADORA3KDM4EMEN1GAA
SCHEMBL28473632 0.74 PARP1 (0.51) MCL1ADORA3KDM4EMEN1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5760191-A Macrocyclic complexing agents and targeting immunoreagents useful in therapeutic and diagnostic compositions and methods NYCOMED IMAGING AS (NO) 1998-06-02 US disclosed