SCHEMBL8701589

SCHEMBL8701589

CCc1ccc2c(c1)NC(=O)C2(CCN1CCC(c2cccc(C(F)(F)F)c2)CC1)c1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 2/20 0.52
HTR7 P34969 3/20 0.43
CHRM4 P08173 1/20 0.42
DRD4 P21917 1/20 0.42
GRM2 Q14416 1/20 0.42
CHRM3 P20309 1/20 0.41
CCR2 P41597 4/20 0.40
NR3C1 P04150 2/20 0.40
TRPV6 Q9H1D0 1/20 0.40
KDM4A O75164 1/20 0.40
KDM4B O94953 1/20 0.40
KDM5C P41229 1/20 0.40
KDM5B Q9UGL1 1/20 0.40
CCR5 P51681 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8706668 0.84 HTR7 (0.57) DRD2HTR7
Hydrochloric Acid SCHEMBL8701973 0.83 HTR7 (0.43) DRD2HTR7
SCHEMBL8702980 0.78 SIGMAR1 (0.44) HTR7
Hydrochloric Acid SCHEMBL8708208 0.78 HTR7 (0.46) DRD2HTR7
SCHEMBL8701565 0.76 HTR7 (0.55) DRD2HTR7
Hydrochloric Acid SCHEMBL8707983 0.76 HTR7 (0.51) DRD2HTR7
Hydrochloric Acid SCHEMBL8706250 0.73 HTR7 (0.52) DRD2HTR7
Hydrochloric Acid SCHEMBL8708209 0.72 HTR7 (0.56) DRD2HTR7DRD4
Hydrochloric Acid SCHEMBL8702092 0.71 HTR7 (0.47) DRD2HTR7
Hydrochloric Acid SCHEMBL8702749 0.71 HTR7 (0.54) DRD2HTR7DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998002432-A1 BICYCLIC COMPOUNDS FOR CONTROLLING MICTURITION TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-01-22 WO disclosed