SCHEMBL8705185

SCHEMBL8705185

COc1ccc(N2CCNCC2)cc1OC(C)=O

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 2/20 0.49
HTR7 P34969 2/20 0.49
ADRB1 P08588 4/20 0.49
HTR3E A5X5Y0 2/20 0.49
HTR3B O95264 2/20 0.49
HTR3A P46098 2/20 0.49
HTR3D Q70Z44 2/20 0.49
HTR3C Q8WXA8 2/20 0.49
SIGMAR1 Q99720 1/20 0.49
ACVR1 Q04771 3/20 0.48
HTR1D P28221 1/20 0.48
HTR1B P28222 1/20 0.48
CHRNB2 P17787 1/20 0.47
CHRNA4 P43681 1/20 0.47
TGFBR1 P36897 2/20 0.47
KDR P35968 1/20 0.46
ALDH1A1 P00352 1/20 0.46
ABCB1 P08183 2/20 0.46
ALK Q9UM73 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL361649 0.85 ADRB1 (0.61) HTR1AHTR7ADRB1HTR3EHTR3B
Hydrochloric Acid SCHEMBL2156292 0.84 ADRB1 (0.59) HTR1AHTR7ADRB1HTR3EHTR3B
Hydrochloric Acid SCHEMBL7711565 0.84 ADRB1 (0.59) HTR1AHTR7ADRB1HTR3EHTR3B
SCHEMBL8257139 0.82 ABCB1 (0.54) HTR1AHTR7ADRB1HTR3EHTR3B
SCHEMBL1107020 0.79 CHRNB2 (0.46) HTR1AHTR7ADRB1HTR3EHTR3B
SCHEMBL2292016 0.78 FYN (0.58) HTR1AHTR7ADRB1HTR3EHTR3B
SCHEMBL1600775 0.78 ADRB1 (0.56) HTR1AHTR7ADRB1HTR3EHTR3B
SCHEMBL8257463 0.78 ABCB1 (0.53) HTR1AHTR7ADRB1HTR3EHTR3B
SCHEMBL19579582 0.78 ACVR1 (0.51) HTR1AHTR7ADRB1HTR3EHTR3B
SCHEMBL873466 0.77 ADRB1 (0.51) HTR1AHTR7ADRB1HTR3EHTR3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5780472-A ANTITUMOR AGENTS SAMJIN PHARMACEUTICAZL CO., LTD. (KR) 1998-07-14 US disclosed
EP-0749425-A1 NEW PIPERAZINE DERIVATIVES AND METHODS FOR THE PREPARATION THEREOF AND COMPOSITIONS CONTAINING THE SAME SAMJIN PHARM. CO., LTD. (KR) 1996-12-27 EP disclosed
WO-1996021648-A1 NEW PIPERAZINE DERIVATIVES AND METHODS FOR THE PREPARATION THEREOF AND COMPOSITIONS CONTAINING THE SAME SAMJIN PHARMACEUTICAL CO., LTD. (KR) 1996-07-18 WO disclosed