SCHEMBL8705209

SCHEMBL8705209

CC(=O)Nc1ccc2c(c1)CC(CCc1nnn[nH]1)C2

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 2/20 0.38
HTR2B P41595 2/20 0.38
CYP1A2 P05177 1/20 0.38
ADRA2A P08913 1/20 0.38
MAOA P21397 1/20 0.38
SLC6A2 P23975 1/20 0.38
SLC6A4 P31645 1/20 0.38
MTNR1A P48039 1/20 0.38
BAZ2B Q9UIF8 1/20 0.38
HTR2A P28223 1/20 0.36
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
ROCK2 O75116 1/20 0.36
ROCK1 Q13464 1/20 0.36
NQO2 P16083 1/20 0.35
CHRNB2 P17787 1/20 0.34
CHRNA4 P43681 1/20 0.34
GRIA2 P42262 1/20 0.34
NAMPT P43490 1/20 0.34
OPRD1 P41143 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8703784 0.89 HTR2C (0.40) HTR2CHTR2BCYP1A2ADRA2AMAOA
SCHEMBL8703648 0.81 CA1 (0.31)
SCHEMBL12355697 0.77 FYN (0.50) HTR2CHTR2BCYP1A2ADRA2AMAOA
SCHEMBL8700156 0.75 IDO1 (0.44) HTR2BADRA2ASLC6A4HTR2A
SCHEMBL12355679 0.74 CYP1A2 (0.50) HTR2CHTR2BCYP1A2ADRA2AMAOA
SCHEMBL8700889 0.74 PNMT (0.44) ADRA2A
SCHEMBL2246016 0.72 CYP1A2 (0.44) HTR2CHTR2BCYP1A2ADRA2AMAOA
SCHEMBL5582685 0.71 MCHR1 (0.54) HTR2CHTR2BCYP1A2ADRA2AMAOA
SCHEMBL2250545 0.70 CYP1A2 (0.46) HTR2CHTR2BCYP1A2ADRA2AMAOA
SCHEMBL2246315 0.69 CYP1A2 (0.54) HTR2CHTR2BCYP1A2ADRA2AMAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998005651-A1 NOVEL GLUTAMATE RECEPTOR ANTAGONISTS: FUSED CYCLOALKYL QUINOXALINEDIONES WARNER-LAMBERT COMPANY (US) 1998-02-12 WO disclosed