SCHEMBL8705259

SCHEMBL8705259

O=C1C=c2cccnc2=CC1=O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S100A4 P26447 3/20 0.38
CDC25B P30305 3/20 0.38
TDP1 Q9NUW8 4/20 0.37
TDP2 O95551 2/20 0.37
NSD2 O96028 2/20 0.37
PAX8 Q06710 2/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
ABL1 P00519 1/20 0.37
PLCG1 P19174 1/20 0.37
CES1 P23141 1/20 0.37
RIN1 Q13671 1/20 0.37
THRB P10828 1/20 0.37
BLM P54132 1/20 0.37
GAA P10253 1/20 0.37
TGM2 P21980 1/20 0.36
PADI1 Q9ULC6 1/20 0.36
PADI3 Q9ULW8 1/20 0.36
PADI4 Q9UM07 1/20 0.36
PADI2 Q9Y2J8 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9728861 0.75 MAPT (0.37) MEN1KMT2AMAPTKDM4ESMN1; SMN2
SCHEMBL9728856 0.75 MAPT (0.37) MEN1KMT2AMAPTKDM4ESMN1; SMN2
SCHEMBL9728849 0.75 MAPT (0.37) MEN1KMT2AMAPTKDM4ESMN1; SMN2
SCHEMBL26924676 0.71 TDP2 (0.32) TDP1TDP2NSD2PAX8MEN1
SCHEMBL18921 0.71 TDP2 (0.32) TDP1TDP2NSD2PAX8MEN1
Hydrochloric Acid SCHEMBL6025175 0.70 TDP2 (0.31) TDP1TDP2NSD2PAX8MEN1
SCHEMBL2230292 0.68 MAPT (0.40) S100A4CDC25BTDP1TDP2NSD2
SCHEMBL28978114 0.68 S100A4 (0.34) S100A4CDC25BTDP1TDP2NSD2
SCHEMBL670066 0.68 BRD4 (0.36) S100A4CDC25BTDP1TDP2NSD2
SCHEMBL4074635 0.66 MAPT (0.39) S100A4CDC25BTDP1TDP2NSD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014071316-A1 IN SILICO IDENTIFICATION OF CANCER MOLECULAR SIGNALING PATHWAYS AND DRUG CANDIDATES H. LEE MOFFITT CANCER CENTER AND RESEARCH INSTITUTE, INC. (US) 2014-05-08 WO disclosed
US-5733918-A ANTITUMOR AGENT TAIHO PHARMACEUTICAL CO., LTD. (JP) 1998-03-31 US disclosed
US-5710162-A ANTITUMOR AGENTS TAIHO PHARMACEUTICAL CO., LTD. (JP) 1998-01-20 US disclosed