SCHEMBL8709202

SCHEMBL8709202

COc1cc2ncnc(CNc3cccc(Cl)c3)c2cc1OC

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 11/20 0.65
MAPK1 P28482 5/20 0.65
KDM4E B2RXH2 3/20 0.65
MAPT P10636 2/20 0.65
RAF1 P04049 2/20 0.65
FBP1 P09467 2/20 0.65
ALDH1A1 P00352 2/20 0.65
MEN1 O00255 1/20 0.65
GMNN O75496 1/20 0.65
ABL1 P00519 1/20 0.65
LMNA P02545 1/20 0.65
TP53 P04637 1/20 0.65
CYP1A2 P05177 1/20 0.65
GLA P06280 1/20 0.65
CYP3A4 P08684 1/20 0.65
CYP2D6 P10635 1/20 0.65
SRC P12931 1/20 0.65
HPGD P15428 1/20 0.65
ALOX15 P16050 1/20 0.65
NFKB1 P19838 1/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8501510 0.99 EGFR (0.66) EGFRMAPK1KDM4EMAPTRAF1
SCHEMBL8708364 0.88 EGFR (0.63) EGFRMAPK1KDM4EMAPTRAF1
Hydrochloric Acid SCHEMBL8503111 0.87 EGFR (0.64) EGFRMAPK1KDM4EMAPTRAF1
SCHEMBL8708372 0.83 EGFR (0.67) EGFRMAPTRAF1KMT2AMAPK14
Hydrochloric Acid SCHEMBL8503039 0.82 EGFR (0.66) EGFRMAPTRAF1MAPK14LCK
SCHEMBL8704642 0.80 HTT (0.62) EGFRMAPK1KDM4EALDH1A1MEN1
Tyrphostin Ag-1478 SCHEMBL31079458 0.79 EGFR (1.00) EGFRMAPK1KDM4EMAPTRAF1
Tyrphostin Ag-1478 SCHEMBL29350062 0.79 EGFR (1.00) EGFRMAPK1KDM4EMAPTRAF1
Tyrphostin Ag-1478 SCHEMBL93838 0.79 EGFR (1.00) EGFRMAPK1KDM4EMAPTRAF1
Tyrphostin Ag-1478 SCHEMBL29483198 0.79 EGFR (1.00) EGFRMAPK1KDM4EMAPTRAF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5710158-A INHIBITORS OF PROTEIN TYROSINE KINASE AND EPIDERMAL GROWTH FACTOR RHONE-POULENC RORER PHARMACEUTICALS INC. (US) 1998-01-20 US claimed