SCHEMBL8709382

SCHEMBL8709382

COc1ccc(NC(=S)C(C)C)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 3/20 0.59
CYP1A2 P05177 3/20 0.58
CYP2C19 P33261 3/20 0.58
MAOA P21397 2/20 0.56
MAOB P27338 2/20 0.56
ALDH1A1 P00352 6/20 0.55
MAPT P10636 5/20 0.55
GAA P10253 3/20 0.55
RAB9A P51151 7/20 0.55
SMN1; SMN2 Q16637 6/20 0.55
NPC1 O15118 6/20 0.55
CYP2C9 P11712 2/20 0.54
CYP2D6 P10635 1/20 0.54
MEN1 O00255 2/20 0.53
KMT2A Q03164 2/20 0.53
HTT P42858 2/20 0.53
LMNA P02545 2/20 0.51
TDP1 Q9NUW8 1/20 0.51
CYP3A4 P08684 1/20 0.50
TP53 P04637 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21325519 0.85 SMN1; SMN2 (0.42) HPGDCYP1A2CYP2C19ALDH1A1MAPT
SCHEMBL8167087 0.79 CYP1A2 (0.85) HPGDCYP1A2CYP2C19MAOAMAOB
SCHEMBL13754514 0.78 ALDH1A1 (0.69) HPGDCYP1A2CYP2C19MAOAMAOB
SCHEMBL13715007 0.78 HPGD (0.66) HPGDCYP1A2CYP2C19MAOAMAOB
SCHEMBL19035711 0.78 SMN1; SMN2 (0.55) HPGDCYP1A2CYP2C19ALDH1A1MAPT
SCHEMBL7306947 0.78 CYP1A2 (0.69) HPGDCYP1A2CYP2C19MAOAMAOB
SCHEMBL3667176 0.77 ALDH1A1 (0.56) HPGDCYP1A2CYP2C19MAOAMAOB
SCHEMBL2608943 0.77 HTT (0.70) HPGDCYP1A2CYP2C19ALDH1A1MAPT
SCHEMBL14519904 0.77 RAB9A (0.55) HPGDCYP1A2CYP2C19MAOAMAOB
SCHEMBL23944962 0.76 MEN1 (0.54) ALDH1A1MAPTGAARAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9687832-B2 Bifunctional organic catalysts OXFORD UNIVERSITY INNOVATION LIMITED (GB) 2017-06-27 US disclosed
CN-1252717-A Intermediate and method for preparing benzo [ b ] thiophene LILLY CO ELI (US) 2000-05-10 CN disclosed
WO-1998048787-A1 INTERMEDIATES AND A PROCESS FOR PREPARING BENZO[b]THIOPHENES ELI LILLY AND COMPANY (US) 1998-11-05 WO disclosed