SCHEMBL8710480

SCHEMBL8710480

O=C(c1c[nH]c2ccccc12)N1CCC(Cc2ccccc2)CC1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 2/20 0.71
MAPK14 Q16539 6/20 0.67
HTT P42858 1/20 0.67
CHRM2 P08172 1/20 0.64
TACR1 P25103 1/20 0.62
TACR3 P29371 1/20 0.62
CYP2C9 P11712 5/20 0.60
CYP2C19 P33261 5/20 0.60
HTR2B P41595 3/20 0.60
GFER P55789 1/20 0.60
TPSAB1 Q15661 1/20 0.57
GRIN2D O15399 1/20 0.56
GRIN3B O60391 1/20 0.56
GRIN1 Q05586 1/20 0.56
GRIN2A Q12879 1/20 0.56
GRIN2C Q14957 1/20 0.56
GRIN3A Q8TCU5 1/20 0.56
GABRA1 P14867 1/20 0.56
GABRG2 P18507 1/20 0.56
GABRB3 P28472 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8707891 0.91 CHRM2 (0.62) GRIN2BMAPK14HTTCHRM2TACR1
SCHEMBL1063370 0.88 MEN1 (0.66) GRIN2BMAPK14HTTCHRM2CYP2C9
SCHEMBL1083550 0.88 MEN1 (0.60) GRIN2BMAPK14HTTCHRM2CYP2C9
SCHEMBL8711840 0.87 MEN1 (0.63) GRIN2BMAPK14CYP2C9CYP2C19HTR2B
SCHEMBL8707900 0.87 MAPK14 (0.60) GRIN2BMAPK14HTTCYP2C9CYP2C19
SCHEMBL8708970 0.87 CYP2C9 (0.60) GRIN2BMAPK14CHRM2CYP2C9CYP2C19
SCHEMBL8707313 0.87 TPSAB1 (0.61) GRIN2BMAPK14CYP2C9CYP2C19HTR2B
SCHEMBL8707626 0.86 TACR1 (0.61) GRIN2BMAPK14HTTCHRM2TACR1
SCHEMBL8707640 0.84 MEN1 (0.65) MAPK14CHRM2CYP2C9CYP2C19HTR2B
SCHEMBL8711792 0.83 HTT (0.68) GRIN2BHTTGABRA1GABRG2GABRB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1975620-A2 Three hybrid assay system GPC Biotech AG (DE) 2008-10-01 EP disclosed
WO-1998028292-A1 NOVEL PIPERIDINE CONTAINING COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 1998-07-02 WO disclosed