SCHEMBL8710876

SCHEMBL8710876

COCOc1cc(OC)c([N+](=O)[O-])cc1C=O

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 10/20 0.55
MAPT P10636 7/20 0.55
KDM4E B2RXH2 2/20 0.55
CYP3A4 P08684 1/20 0.55
ALOX15 P16050 1/20 0.55
PRKDC P78527 1/20 0.55
HSD17B10 Q99714 1/20 0.55
TDP1 Q9NUW8 3/20 0.45
TSHR P16473 1/20 0.45
ERN1 O75460 2/20 0.43
LMNA P02545 4/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
HPGD P15428 2/20 0.41
HTT P42858 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
THRB P10828 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3847699 0.86 ALDH1A1 (0.67) ALDH1A1MAPTKDM4ECYP3A4ALOX15
SCHEMBL5338041 0.81 ALDH1A1 (0.68) ALDH1A1MAPTKDM4ECYP3A4ALOX15
SCHEMBL19331554 0.80 ALDH1A1 (0.77) ALDH1A1MAPTKDM4ECYP3A4ALOX15
SCHEMBL20783154 0.79 ALDH1A1 (0.61) ALDH1A1MAPTKDM4ECYP3A4ALOX15
SCHEMBL29125349 0.77 ALDH1A1 (0.63) ALDH1A1MAPTKDM4ECYP3A4ALOX15
SCHEMBL28704679 0.77 ALDH1A1 (0.55) ALDH1A1MAPTKDM4ECYP3A4ALOX15
SCHEMBL8071562 0.77 ALDH1A1 (0.59) ALDH1A1MAPTKDM4ECYP3A4ALOX15
SCHEMBL2723326 0.77 ALDH1A1 (0.83) ALDH1A1MAPTKDM4ECYP3A4ALOX15
SCHEMBL25380949 0.77 ALDH1A1 (0.43) ALDH1A1MAPTKDM4ECYP3A4ALOX15
SCHEMBL8946170 0.76 ALDH1A1 (0.61) ALDH1A1MAPTKDM4ECYP3A4ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5716971-A FOR TREATMENT OF ANGINA PECTORIS AND HYPERTENSION TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-02-10 US disclosed
EP-0623597-B1 Pyridine derivatives, with potassium channel opening activity TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1997-10-22 EP disclosed
EP-0623597-A1 Pyridine derivatives, with potassium channel opening activity Takeda Chemical Industries, Ltd. (JP) 1994-11-09 EP disclosed