SCHEMBL8712707

SCHEMBL8712707

C=C(Cc1ccc(OC(C)C)c(Br)c1)[N+](=O)[O-]

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 5/20 0.39
HDAC6 Q9UBN7 2/20 0.39
PDK1 Q15118 1/20 0.37
ABL1 P00519 1/20 0.36
RIN1 Q13671 1/20 0.36
S1PR3 Q99500 1/20 0.35
S1PR5 Q9H228 1/20 0.35
RXRA P19793 1/20 0.35
RXRB P28702 1/20 0.35
RXRG P48443 1/20 0.35
CSNK2A1 P68400 2/20 0.35
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
XDH P47989 1/20 0.34
POLB P06746 1/20 0.33
LMNA P02545 1/20 0.33
ATM Q13315 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
HTR2A P28223 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8709313 0.85 HDAC1 (0.53) HDAC1HDAC6ABL1RIN1KDM4E
SCHEMBL8388481 0.77 POLB (0.57) HDAC1HDAC6ABL1RIN1S1PR3
SCHEMBL8712614 0.75 ABL1 (0.42) HDAC1HDAC6ABL1RIN1S1PR3
SCHEMBL3719650 0.75 CSNK2A1 (0.45) ABL1RIN1S1PR3S1PR5RXRA
SCHEMBL8867113 0.75 LMNA (0.49) ALDH1A1LMNASMN1; SMN2
SCHEMBL15057261 0.73 ABL1 (0.49) HDAC1HDAC6ABL1RIN1S1PR3
SCHEMBL3723071 0.72 CSNK2A1 (0.45) S1PR3S1PR5RXRARXRBRXRG
SCHEMBL11148098 0.71 HTT (0.43) KDM4EALDH1A1LMNASMN1; SMN2
SCHEMBL8113158 0.71 CYP19A1 (0.54) PDK1ALDH1A1TDP1LMNASMN1; SMN2
SCHEMBL28293124 0.70 CSNK2A1 (0.65) S1PR3S1PR5CSNK2A1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998017660-A1 PHENYL SPIROETHERCYCLOALKYL TACHYKININ RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 1998-04-30 WO disclosed