SCHEMBL8713164

SCHEMBL8713164

COCOCOC.Oc1ccc(C=C(Br)Br)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 3/20 0.41
ESR2 Q92731 3/20 0.41
PTGS2 P35354 3/20 0.41
NQO2 P16083 2/20 0.41
PTGS1 P23219 2/20 0.41
KDM4E B2RXH2 2/20 0.39
ALDH1A1 P00352 1/20 0.39
ABCG2 Q9UNQ0 2/20 0.37
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
THRB P10828 1/20 0.36
CISD1 Q9NZ45 1/20 0.36
BACE1 P56817 2/20 0.36
TTR P02766 2/20 0.36
CYP1A1 P04798 2/20 0.36
ALOX5 P09917 2/20 0.36
CYP1B1 Q16678 2/20 0.36
CA12 O43570 2/20 0.36
CA1 P00915 2/20 0.36
CA2 P00918 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8713174 0.83 ESR1 (0.47) ESR1ESR2PTGS2NQO2PTGS1
SCHEMBL3754984 0.80 ESR1 (0.54) ESR1ESR2PTGS2NQO2PTGS1
4-Hydroxybenzaldehyde SCHEMBL9157915 0.78 ALDH5A1 (0.61) KDM4EALDH1A1BACE1CA12CA1
SCHEMBL8713169 0.76 MAPT (0.39) ESR1PTGS2NQO2PTGS1KDM4E
Phenol SCHEMBL11804127 0.70 CA4 (0.52) ESR1ESR2PTGS2PTGS1ALDH1A1
4-Hydroxybenzaldehyde SCHEMBL28883554 0.69 ALDH5A1 (0.67) PTGS2NQO2PTGS1KDM4EALDH1A1
SCHEMBL8709934 0.69 ALDH1A1 (0.48) ESR1ESR2PTGS2PTGS1KDM4E
SCHEMBL15452321 0.69 IDO1 (0.48) ESR1ESR2KDM4EALDH1A1MEN1
SCHEMBL1164737 0.69 ALDH1A1 (0.61) PTGS2NQO2PTGS1KDM4EALDH1A1
SCHEMBL7095950 0.68 ESR1 (0.48) ESR1ESR2PTGS2NQO2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5716971-A FOR TREATMENT OF ANGINA PECTORIS AND HYPERTENSION TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-02-10 US disclosed
EP-0623597-B1 Pyridine derivatives, with potassium channel opening activity TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1997-10-22 EP disclosed
EP-0623597-A1 Pyridine derivatives, with potassium channel opening activity Takeda Chemical Industries, Ltd. (JP) 1994-11-09 EP disclosed