SCHEMBL8713428

SCHEMBL8713428

O=C(Cl)c1nn(CC2CC2)c2ccccc12

nearest known ligand 0.52

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 3/20 0.52
CNR2 P34972 2/20 0.47
ACHE P22303 1/20 0.47
SSTR4 P31391 1/20 0.47
ROCK2 O75116 3/20 0.45
HTR4 Q13639 1/20 0.44
HTR3A P46098 8/20 0.44
PADI4 Q9UM07 1/20 0.43
USP30 Q70CQ3 1/20 0.43
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
TSHR P16473 1/20 0.41
PMP22 Q01453 1/20 0.41
HIF1A Q16665 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31429317 0.87 CNR1 (0.53) CNR1CNR2ACHESSTR4ROCK2
SCHEMBL8719218 0.87 CNR1 (0.53) CNR1CNR2ACHESSTR4ROCK2
SCHEMBL5433258 0.86 CNR1 (0.57) CNR1CNR2ACHESSTR4PADI4
SCHEMBL31429457 0.82 CNR1 (0.54) CNR1CNR2ACHESSTR4ROCK2
SCHEMBL24437187 0.82 CNR1 (0.56) CNR1CNR2ACHESSTR4ROCK2
SCHEMBL31429426 0.82 CNR1 (0.56) CNR1CNR2ACHESSTR4ROCK2
SCHEMBL4052657 0.81 CNR1 (0.61) CNR1CNR2ACHESSTR4ROCK2
SCHEMBL6950019 0.79 CYP1A2 (0.45) CNR1CNR2SSTR4HTR3ACYP1A2
SCHEMBL15882181 0.79 HTR4 (0.48) CNR1CNR2ACHEROCK2HTR4
SCHEMBL31429308 0.79 HTR4 (0.48) CNR1CNR2ACHEROCK2HTR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0708105-B1 5-HT4 receptor agonists NISSHIN FLOUR MILLING CO (JP) 1998-12-23 EP disclosed
US-5684003-A GASTROINTESTINAL DISORDERS OR ANTIULCER AGENTS NISSHIN FLOUR MILLING CO., LTD. (JP) 1997-11-04 US disclosed
EP-0708105-A1 5-HT4 receptor agonists NISSHIN FLOUR MILLING CO., LTD. (JP) 1996-04-24 EP disclosed