SCHEMBL8714007

SCHEMBL8714007

O=S(=O)(O)CCC(O)(c1ccccc1)N(Cc1ccccc1)Cc1ccccc1

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CA2 P00918 1/20 0.38
RORC P51449 1/20 0.36
CYP2C9 P11712 2/20 0.36
CYP2C19 P33261 2/20 0.36
CYP1A2 P05177 1/20 0.36
RIPK1 Q13546 2/20 0.35
NR1H3 Q13133 2/20 0.35
PTPN1 P18031 1/20 0.35
HSD11B1 P28845 1/20 0.34
NR1H2 P55055 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
TAS2R14 Q9NYV8 1/20 0.34
CYP2D6 P10635 2/20 0.33
TSHR P16473 1/20 0.33
LTA4H P09960 1/20 0.33
MAPK1 P28482 1/20 0.33
SERPINE1 P05121 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL353290 0.70 OPRM1 (0.42) CA2RORCRIPK1MEN1KMT2A
SCHEMBL8504022 0.69 ALDH1A1 (0.40) CA2CYP2C9CYP2C19CYP1A2HSD11B1
SCHEMBL22861240 0.68 CA2 (0.46) CA2HSD11B1MEN1KMT2ATAS2R14
SCHEMBL16680276 0.68 CYP1A2 (0.41) CA2CYP2C9CYP2C19CYP1A2PTPN1
SCHEMBL22861236 0.68 HDAC3 (0.46) CA2RORCHSD11B1MEN1KMT2A
SCHEMBL10655752 0.68 TSHR (0.50) CA2CYP2C19NR1H3NR1H2CYP2D6
SCHEMBL4459190 0.67 CA2 (0.48) CA2HSD11B1MEN1KMT2ATAS2R14
SCHEMBL918029 0.66 HDAC3 (0.51) CA2RORCLTA4H
SCHEMBL27273867 0.66 HDAC3 (0.47) CA2RORCLTA4H
SCHEMBL28523868 0.66 CA2 (0.43) CA2HSD11B1MEN1KMT2ATAS2R14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0861233-A1 N-PROTECTED/N-SUBSTITUTED-BETA-AMINO HYDROXY SULFONATES G.D. SEARLE & CO. (US) 1998-09-02 EP claimed
WO-1997018190-A1 N-PROTECTED/N-SUBSTITUTED-BETA-AMINO HYDROXY SULFONATES G.D. SEARLE & CO. (US) 1997-05-22 WO claimed
EP-0861233-A1 N-PROTECTED/N-SUBSTITUTED-BETA-AMINO HYDROXY SULFONATES G.D. SEARLE & CO. (US) 1998-09-02 EP disclosed
WO-1997018190-A1 N-PROTECTED/N-SUBSTITUTED-BETA-AMINO HYDROXY SULFONATES G.D. SEARLE & CO. (US) 1997-05-22 WO disclosed