Leucine

Leucine

SCHEMBL8714828

CB(O)O.CC(C)C[C@H](N)C(=O)O.C[C@@H](C(=O)O)N(C(=O)N1CCOCC1)c1cccc2ccccc12

nearest known ligand 0.37

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.37
KDM4E B2RXH2 4/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
MAPT P10636 1/20 0.37
TSHR P16473 1/20 0.37
HSD17B10 Q99714 1/20 0.37
NPC1 O15118 2/20 0.36
RAB9A P51151 1/20 0.36
MMP2 P08253 1/20 0.35
MMP9 P14780 1/20 0.35
MMP8 P22894 1/20 0.35
HTT P42858 1/20 0.35
LMNA P02545 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
CNR1 P21554 2/20 0.35
HTR2C P28335 1/20 0.35
CNR2 P34972 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
GRIK1 P39086 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL901425 0.90 ALDH1A1 (0.38) ALDH1A1KDM4ESMN1; SMN2MAPTTSHR
SCHEMBL6799660 0.86 ALDH1A1 (0.47) ALDH1A1KDM4ESMN1; SMN2MAPTTSHR
Mannitol SCHEMBL7620660 0.79 CASR (0.34) ALDH1A1KDM4ESMN1; SMN2MAPTTSHR
Leucine SCHEMBL2297615 0.77 MMP2 (0.49) ALDH1A1KDM4ETSHRHSD17B10MMP2
SCHEMBL7289294 0.76 ALDH1A1 (0.52) ALDH1A1KDM4ESMN1; SMN2MAPTTSHR
Leucine SCHEMBL3812226 0.74 MMP2 (0.48) ALDH1A1KDM4ETSHRHSD17B10MMP2
Leucine SCHEMBL1406254 0.72 MMP2 (0.50) ALDH1A1KDM4ETSHRHSD17B10MMP2
SCHEMBL8713936 0.72 KDM4E (0.36) ALDH1A1KDM4ESMN1; SMN2MAPTTSHR
SCHEMBL6801153 0.71 ALDH1A1 (0.49) ALDH1A1SMN1; SMN2TSHRHSD17B10LMNA
Leucine SCHEMBL28593704 0.70 SLC7A5 (0.40) GRIK1GRIK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0788360-A4 BORONIC ESTER AND ACID COMPOUNDS, SYNTHESIS AND USES PROSCRIPT INC (US) 1998-05-06 EP disclosed
EP-0788360-A1 BORONIC ESTER AND ACID COMPOUNDS, SYNTHESIS AND USES PROSCRIPT, INC. (US) 1997-08-13 EP disclosed